SCHEMBL4874161

SCHEMBL4874161

Nc1ccccc1C(=O)c1ccc2c(c1)NC(=O)C2

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 3/20 0.51
HDAC3 O15379 2/20 0.51
HDAC1 Q13547 1/20 0.51
CRBN Q96SW2 2/20 0.50
GAA P10253 2/20 0.47
MAPT P10636 1/20 0.47
AHR P35869 3/20 0.45
HSD11B1 P28845 2/20 0.45
PDK2 Q15119 1/20 0.45
CMA1 P23946 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
EIF2AK2 P19525 1/20 0.43
HDAC6 Q9UBN7 1/20 0.40
TDP2 O95551 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874148 0.86 SMYD3 (0.51) SMYD3HDAC3HDAC1CRBNGAA
SCHEMBL7679044 0.81 SMYD3 (0.53) SMYD3HDAC3HDAC1CRBNGAA
SCHEMBL3573881 0.80 SMYD3 (0.55) SMYD3HDAC3HDAC1CRBNAHR
SCHEMBL3578248 0.80 SMYD3 (0.52) SMYD3HDAC3HDAC1CRBNAHR
SCHEMBL3573876 0.79 SMYD3 (0.56) SMYD3HDAC3HDAC1CRBNAHR
SCHEMBL6543874 0.78 FADS1 (0.50) HDAC3HDAC1
SCHEMBL3581639 0.78 TDP2 (0.55) SMYD3HDAC3HDAC1CRBNAHR
SCHEMBL3194345 0.78 SMYD3 (0.58) SMYD3HDAC3HDAC1CRBNAHR
SCHEMBL30760741 0.78 SMYD3 (0.58) SMYD3HDAC3HDAC1CRBNAHR
Hydrochloric Acid SCHEMBL29528151 0.76 SMYD3 (0.57) SMYD3HDAC3HDAC1CRBNAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902025-A1 KINASE INHIBITORS Allergan, Inc. (US) 2008-03-26 EP disclosed
WO-2007008895-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2007-01-18 WO disclosed