SCHEMBL4874499

SCHEMBL4874499

O=C(c1ccc(=O)n(-c2c(Cl)cccc2Cl)c1)c1ccc(F)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
RORC P51449 3/20 0.42
HSD11B1 P28845 1/20 0.41
NPC1 O15118 1/20 0.41
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
HPGD P15428 1/20 0.39
P2RX7 Q99572 3/20 0.38
SRD5A2 P31213 1/20 0.36
CDK2 P24941 1/20 0.36
PYGL P06737 1/20 0.36
CYP2D6 P10635 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4877819 0.91 MAPK14 (0.49) RORCMAPK13MAPK12MAPK11MAPK14
SCHEMBL4924074 0.90 MAPK14 (0.41) ALDH1A1RORCNPC1MAPK13MAPK12
SCHEMBL4877829 0.84 HSD11B1 (0.37) RORCHSD11B1KDM4EPOLBMAPK13
SCHEMBL4877832 0.84 HSD11B1 (0.37) RORCHSD11B1KDM4EPOLBMAPK13
SCHEMBL4917597 0.82 THRB (0.39) LMNARORCNPC1MAPK13MAPK12
SCHEMBL4878352 0.81 MAPK14 (0.35) ALDH1A1RORCHSD11B1KDM4EPOLB
SCHEMBL4878366 0.81 MAPK14 (0.35) ALDH1A1RORCHSD11B1KDM4EPOLB
SCHEMBL375227 0.80 TP53 (0.41) ALDH1A1LMNAKDM4EHPGDP2RX7
SCHEMBL4877345 0.80 MAPK14 (0.42) ALDH1A1LMNAGAAPKMRORC
SCHEMBL4876312 0.79 MAPK14 (0.39) RORCMAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080081825-A1 Nitrogen-Containing Heterocyclic Compounds and Medicinal Use Thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2008-04-03 US disclosed
EP-1741702-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2007-01-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080081825-A1 Nitrogen-Containing Heterocyclic Compounds and Medicinal Use Thereof MAPK1, NOS1, NOS2 ALDH1A1 1539/4885LMNA 2177/4885GAA 2432/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.