SCHEMBL4874928

SCHEMBL4874928

C[C@@H](C(=O)O)n1c(Cl)cc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.42
KMT2A Q03164 3/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
DAO P14920 1/20 0.40
CCR2 P41597 3/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
KDM4E B2RXH2 3/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NTSR1 P30989 1/20 0.36
GAA P10253 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037330 0.82 KMT2A (0.46) MCL1KMT2ADAOALDH1A1TSHR
SCHEMBL6287877 0.77 HTR4 (0.41) MCL1KMT2ADAOKDM4EGAA
SCHEMBL21359462 0.76 OXER1 (0.46) MCL1ALDH1A1
SCHEMBL6286028 0.73 HTR4 (0.38) MCL1KMT2ADAOALDH1A1HPGD
SCHEMBL6286022 0.73 HTR4 (0.38) MCL1KMT2ADAOALDH1A1HPGD
SCHEMBL11397353 0.73 ALDH1A1 (0.41) KMT2APTGDR2ALDH1A1TSHRKDM4E
SCHEMBL18258624 0.72 KMT2A (0.53) KMT2AALDH1A1KDM4EMEN1HTT
SCHEMBL18180382 0.72 KMT2A (0.45) KMT2AKDM4EGAACASP1CASP7
SCHEMBL150034 0.72 KMT2A (0.53) KMT2AALDH1A1KDM4EMEN1HTT
SCHEMBL3842692 0.70 DAO (0.46) MCL1KMT2ADAOCCR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963281-A2 HETEROCYCLIC DERIVATIVES AS MODULATORS OF ION CHANNELS Vertex Pharmaceuticals, Inc. (US) 2008-09-03 EP disclosed
WO-2007075895-A2 HETEROCYCLIC DERIVATIVES AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-07-05 WO disclosed