SCHEMBL4877141

SCHEMBL4877141

O=C(O)c1cc2c(s1)c(-c1ccccc1)c(-c1ccc3nc(-c4ccccc4Cl)ccc3c1)n2CC(=O)N1CCC(O)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.36
MAPT P10636 3/20 0.36
HTT P42858 3/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
ABL1 P00519 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SMO Q99835 1/20 0.34
EIF4E P06730 1/20 0.33
HTR2C P28335 1/20 0.33
NPY5R Q15761 2/20 0.33
HSD11B1 P28845 1/20 0.33
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4877132 0.90 MAPT (0.35) LMNAMAPTHTTALDH1A1POLB
SCHEMBL4878306 0.89 PIK3CA (0.40) LMNAMAPTHTTSMOPIK3CA
SCHEMBL4877128 0.88 LMNA (0.36) LMNAALDH1A1POLBKMT2ASMN1; SMN2
SCHEMBL4875677 0.88 GRIN2B (0.34) LMNAMAPTALDH1A1KMT2ASMN1; SMN2
SCHEMBL4878029 0.88 SMO (0.34) LMNAMAPTHTTALDH1A1POLB
SCHEMBL4866875 0.86 ALDH1A1 (0.39) LMNAMAPTALDH1A1POLBMEN1
SCHEMBL4872104 0.86 KDM4E (0.40) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL4877312 0.86 PIK3CA (0.43) LMNAMAPTHTTALDH1A1MEN1
SCHEMBL4868321 0.86 KCNH2 (0.38) LMNASMOPIK3CAMTOR
SCHEMBL4879113 0.85 GRIN2B (0.34) LMNASMOPIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080051384-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. 2008-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080051384-A1 ANTIVIRAL AGENTS EIF2AK2, MAVS, ZC3HAV1 LMNA 3337/4885MAPT 4372/4885HTT 4667/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.