SCHEMBL488233

SCHEMBL488233

CC1(C)OB(c2cccc(NS(=O)(=O)CCN3CCOCC3)c2)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
EPHX2 P34913 4/20 0.39
TSHR P16473 1/20 0.39
MAP4K4 O95819 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
RECQL P46063 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488274 0.91 SRC (0.44) MAP4K4ALDH1A1CA12CA1CA2
SCHEMBL488893 0.90 SRC (0.44) MEN1KMT2AMAP4K4ALDH1A1CA12
SCHEMBL488839 0.87 CA1 (0.52) MEN1KMT2AEPHX2TSHRMAP4K4
SCHEMBL488765 0.87 KDM1A (0.40) MEN1KMT2ACA12CA1CA2
SCHEMBL488629 0.86 SMN1; SMN2 (0.38) EPHX2CA12CA1CA2CA3
SCHEMBL17896410 0.84 MAP4K4 (0.48) MEN1KMT2AEPHX2MAP4K4CYP3A4
SCHEMBL488672 0.84 ROCK1 (0.36) CA12CA1CA2CA3CA4
SCHEMBL488764 0.83 CYP2D6 (0.38) CA12CA1CA2CA3CA4
SCHEMBL2508131 0.81 LPL (0.48) MEN1KMT2ACA12CA1CA2
SCHEMBL16238072 0.79 LPL (0.48) CA12CA1CA2CA3CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed