SCHEMBL488629

SCHEMBL488629

CC(=O)N1CCN(CCS(=O)(=O)Nc2cccc(B3OC(C)(C)C(C)(C)O3)c2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
KDM1A O60341 3/20 0.37
EPHX2 P34913 5/20 0.36
PARP1 P09874 1/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
SRC P12931 1/20 0.35
ROCK1 Q13464 1/20 0.35
CA12 O43570 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA14 Q9ULX7 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
THRB P10828 2/20 0.34
LOX P28300 1/20 0.34
SLC2A2 P11168 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488672 0.90 ROCK1 (0.36) SMN1; SMN2KDM1APARP1CA1CA2
SCHEMBL488793 0.88 CA1 (0.48) SMN1; SMN2KDM1APARP1CA1CA2
SCHEMBL488274 0.88 SRC (0.44) SMN1; SMN2KDM1APARP1CA1CA2
SCHEMBL488893 0.87 SRC (0.44) SMN1; SMN2KDM1ACA1CA2CA9
SCHEMBL488233 0.86 MEN1 (0.40) EPHX2CA1CA2CA9SRC
SCHEMBL488765 0.85 KDM1A (0.40) KDM1APARP1CA1CA2CA9
SCHEMBL488764 0.82 CYP2D6 (0.38) KDM1ACA1CA2CA9SRC
SCHEMBL488906 0.78 CA1 (0.46) KDM1APARP1CA1CA2CA9
SCHEMBL2508131 0.77 LPL (0.48) SMN1; SMN2CA1CA2CA9CA12
SCHEMBL488724 0.77 PARP1 (0.37) SMN1; SMN2PARP1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed