SCHEMBL488672

SCHEMBL488672

CC1(C)OB(c2cccc(NS(=O)(=O)CCN3CCN(C(=O)CO)CC3)c2)OC1(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.36
PARP1 P09874 1/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
SRC P12931 2/20 0.35
ALK Q9UM73 1/20 0.34
CA12 O43570 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
KDR P35968 2/20 0.33
PDGFRB P09619 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488629 0.90 SMN1; SMN2 (0.38) ROCK1PARP1CA1CA2CA9
SCHEMBL488906 0.88 CA1 (0.46) ROCK1PARP1CA1CA2CA9
SCHEMBL488274 0.86 SRC (0.44) PARP1CA1CA2CA9SRC
SCHEMBL488893 0.85 SRC (0.44) CA1CA2CA9SRCCA12
SCHEMBL488233 0.84 MEN1 (0.40) CA1CA2CA9SRCCA12
SCHEMBL488765 0.83 KDM1A (0.40) PARP1CA1CA2CA9SRC
SCHEMBL488764 0.80 CYP2D6 (0.38) CA1CA2CA9SRCCA12
SCHEMBL488793 0.78 CA1 (0.48) PARP1CA1CA2CA9CA12
SCHEMBL488724 0.77 PARP1 (0.37) PARP1CA1CA2CA9CA12
SCHEMBL2508131 0.76 LPL (0.48) CA1CA2CA9CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed