SCHEMBL488259

SCHEMBL488259

CC(Oc1cccnc1NBr)c1cccc(F)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MET P08581 5/20 0.46
SCN1A P35498 7/20 0.38
SCN5A Q14524 7/20 0.38
SCN8A Q9UQD0 7/20 0.38
GRM5 P41594 1/20 0.38
JAK2 O60674 4/20 0.36
SRC P12931 2/20 0.35
KDR P35968 2/20 0.35
KIT P10721 1/20 0.35
FGFR2 P21802 1/20 0.35
AXL P30530 1/20 0.35
FLT3 P36888 1/20 0.35
MST1R Q04912 1/20 0.35
ALK Q9UM73 2/20 0.34
ROS1 P08922 1/20 0.34
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391902 0.82 MET (0.69) METJAK2SRCKDRKIT
SCHEMBL488617 0.71 MET (0.69) METJAK2ALK
SCHEMBL30453715 0.71 MET (0.69) METJAK2ALK
SCHEMBL15779201 0.65 MET (0.88) METJAK2SRCKDRKIT
SCHEMBL31521440 0.64 ALKBH1 (0.40) METSRCKDRKITFGFR2
SCHEMBL9967747 0.63 GABRA1 (0.44)
SCHEMBL3120131 0.62 MET (1.00) METJAK2SRCKDRKIT
SCHEMBL29529122 0.62 MET (1.00) METJAK2SRCKDRKIT
SCHEMBL488751 0.62 MET (1.00) METJAK2SRCKDRKIT
SCHEMBL15133818 0.62 MET (1.00) METJAK2SRCKDRKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed
US-20070072874-A1 Aminoheteroaryl compounds as protein kinase inhibitors SUGEN, INC. 2007-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072874-A1 Aminoheteroaryl compounds as protein kinase inhibitors MET, MAP4K1, MAP4K2 MET 1/4885SCN1A 1683/4885SCN5A 1586/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.