Cloprednol

Cloprednol

SCHEMBL4886

C[C@]12C=CC(=O)C=C1C(Cl)=C[C@@H]1[C@@H]2[C@@H](O)C[C@@]2(C)[C@H]1CC[C@]2(O)C(=O)CO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 7/20 1.00
NR3C1 P04150 7/20 1.00
NR1I2 O75469 2/20 1.00
MLNR O43193 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
HTR2C P28335 1/20 1.00
HIF1A Q16665 8/20 0.61
HSD17B10 Q99714 8/20 0.61
CYP3A4 P08684 5/20 0.61
CYP2C19 P33261 3/20 0.61
ABCB11 O95342 2/20 0.61
SERPINA6 P08185 2/20 0.61
NR3C2 P08235 2/20 0.61
AR P10275 2/20 0.61
TNF P01375 1/20 0.61
IL6 P05231 1/20 0.61
GLUL P15104 1/20 0.61
ADAM17 P78536 1/20 0.61
GPBAR1 Q8TDU6 1/20 0.61
ALDH1A1 P00352 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cloprednol SCHEMBL19327143 1.00 PGR (1.00) PGRNR3C1NR1I2MLNRADORA3
Cloprednol SCHEMBL11209368 1.00 PGR (1.00) PGRNR3C1NR1I2MLNRADORA3
Cloprednol SCHEMBL25308351 0.97 PGR (0.95) PGRNR3C1NR1I2MLNRADORA3
SCHEMBL11853459 0.90 PGR (0.81) PGRNR3C1NR1I2MLNRADORA3
SCHEMBL11853469 0.90 PGR (0.81) PGRNR3C1NR1I2MLNRADORA3
SCHEMBL11860993 0.89 PGR (0.80) PGRNR3C1NR1I2MLNRADORA3
SCHEMBL11860982 0.89 PGR (0.80) PGRNR3C1NR1I2MLNRADORA3
Cloprednol SCHEMBL3999177 0.84 NR3C1 (0.71) PGRNR3C1NR1I2MLNRADORA3
SCHEMBL11202047 0.83 PGR (0.70) PGRNR3C1NR1I2MLNRADORA3
SCHEMBL11202042 0.83 PGR (0.70) PGRNR3C1NR1I2MLNRADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7326 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
EP-4683679-A1 METHOD FOR DIAGNOSING AND TREATING NIS-EXPRESSING CARCINOMAS AND METASTASES NUSKE, Andreas (DE) 2026-01-28 EP claimed
EP-4301343-B1 PHARMACEUTICAL COMPOSITIONS WITH REDUCED SIDE EFFECT AND METHODS OF USING THE SAME TLC BIOPHARMACEUTICALS INC (US) 2025-11-19 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-20250205227-A1 METHODS FOR ADMINISTERING CORTICOSTEROIDS SPARROW PHARMACEUTICALS, INC. 2025-06-26 US claimed
WO-2025123147-A1 TOLERIZING IMMUNOMODULATORY COMBINATION INTEGRATED NANOTHERAPEUTICS INC. (CA) 2025-06-19 WO claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
US-20250144021-A1 GEL FORMULATIONS FOR LOCAL DRUG RELEASE TECHNICAL UNIVERSITY OF DENMARK (DK) 2025-05-08 US claimed
WO-2025076059-A1 ROCAGLATE DERIVATIVES AND USES THEREOF TRUSTEES OF BOSTON UNIVERSITY (US) 2025-04-10 WO claimed
EP-3943073-B1 BIODEGRADABLE POLYMER MICROPARTICLE CONTAINING STEROID-BASED DRUG AND PREPARATION METHOD THEREFOR REGENBIOTECH INC (KR) 2025-03-26 EP claimed
EP-0173478-B1 Treatment of skin disorders SCOTIA HOLDINGS PLC (GB) 1994-02-02 EP claimed
EP-0540751-A1 STEROID COMPOUND COMBINED WITH POLYSACCHARIDE Eisai Co., Ltd. (JP) 1993-05-12 EP claimed
US-5192528-A Encapsulated in liposomes, aerosols LIPOSOME TECHNOLOGY, INC. (US) 1993-03-09 US claimed
EP-0496520-A1 Novel bone acting agents MERCK & CO. INC. (US) 1992-07-29 EP claimed
US-5049389-A Non-phospholipd lipid, delivery by inhalation LIPOSOME TECHNOLOGY, INC. (US) 1991-09-17 US claimed
US-5043165-A Cholesterol and salt; antiallergens, antiinflammatory agents, skin disorders LIPOSOME TECHNOLOGY, INC. (US) 1991-08-27 US claimed
WO-1990006775-A1 A NOVEL NONPHOSPHOLIPID LIPOSOME COMPOSITION FOR SUSTAINED RELEASE OF DRUGS LIPOSOME TECHNOLOGY, INC. (US) 1990-06-28 WO claimed
US-4906476-A Novel liposome composition for sustained release of steroidal drugs in lungs LIPOSOME TECHNOLOGY, INC. 1990-03-06 US claimed
EP-0173478-A1 Treatment of skin disorders SCOTIA HOLDINGS PLC (GB) 1986-03-05 EP claimed
US-4051241-A ANTIALLERGIC AGENTS, ANTIRHEUMATIC AGENTS, DERMATOLOGIC DRUGS ION SYNTEX (U.S.A.) INC. (US) 1977-09-27 US claimed