SCHEMBL4889158

SCHEMBL4889158

CN1CCN(c2cccc3[nH]c(CNC4CCc5cccnc54)nc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.53
CXCR4 P61073 4/20 0.42
CYP2D6 P10635 1/20 0.42
SLC40A1 Q9NP59 5/20 0.42
BRD4 O60885 1/20 0.38
WNT1 P04628 1/20 0.38
TGFBR1 P36897 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
OPRL1 P41146 1/20 0.38
KCNH2 Q12809 1/20 0.38
DRD4 P21917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4878573 0.94 HTR6 (0.51) HTR6CXCR4CYP2D6SLC40A1KCNH2
SCHEMBL4889721 0.94 HTR6 (0.50) HTR6CXCR4CYP2D6SLC40A1KCNH2
SCHEMBL14270231 0.85 CXCR4 (0.42) CXCR4CYP2D6SLC40A1OPRL1KCNH2
SCHEMBL27889942 0.82 HDAC1 (0.46) CXCR4KCNH2
SCHEMBL4881639 0.81 CXCR4 (0.52) HTR6CXCR4KCNH2
SCHEMBL14270246 0.79 CXCR4 (0.44) CXCR4CYP2D6SLC40A1KCNH2
SCHEMBL4166431 0.79 CXCR4 (0.60) HTR6CXCR4CYP2D6KCNH2DRD4
SCHEMBL4170853 0.79 CXCR4 (0.60) HTR6CXCR4CYP2D6KCNH2DRD4
SCHEMBL5548249 0.79 CXCR4 (0.60) HTR6CXCR4CYP2D6KCNH2DRD4
SCHEMBL13875216 0.79 CXCR4 (0.60) HTR6CXCR4CYP2D6KCNH2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080045537-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-02-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045537-A1 Chemical Compounds CCR5, CXCR4, CXCR3 HTR6 2334/4885CXCR4 2/4885CYP2D6 4070/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.