SCHEMBL4878573

SCHEMBL4878573

CN1CCN(c2cccc3[nH]c(CN[C@H]4CCCc5cccnc54)nc23)CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.51
CXCR4 P61073 15/20 0.46
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CYP2D6 P10635 2/20 0.41
SLC40A1 Q9NP59 1/20 0.41
KCNH2 Q12809 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CYP3A4 P08684 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4889721 0.97 HTR6 (0.50) HTR6CXCR4HDAC1HDAC6CYP2D6
SCHEMBL4889158 0.94 HTR6 (0.53) HTR6CXCR4CYP2D6SLC40A1KCNH2
SCHEMBL27889942 0.88 HDAC1 (0.46) CXCR4HDAC1HDAC6KCNH2
SCHEMBL4878647 0.83 CXCR4 (0.44) HTR6CXCR4CYP2D6KCNH2CHRM2
SCHEMBL14270246 0.83 CXCR4 (0.44) CXCR4HDAC1HDAC6CYP2D6SLC40A1
SCHEMBL4881658 0.82 CXCR4 (0.60) CXCR4KCNH2
SCHEMBL4880484 0.82 CXCR4 (0.60) CXCR4KCNH2
SCHEMBL4889717 0.82 CXCR4 (0.60) CXCR4KCNH2
SCHEMBL4884724 0.81 CXCR4 (0.43) HTR6CXCR4CYP2D6KCNH2CHRM2
SCHEMBL4886423 0.81 CXCR4 (0.58) CXCR4CYP2D6KCNH2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080045537-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-02-21 US disclosed
EP-1789045-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-30 EP disclosed
WO-2006023400-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045537-A1 Chemical Compounds CCR5, CXCR4, CXCR3 HTR6 2334/4885CXCR4 2/4885HDAC1 844/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.