SCHEMBL4890265

SCHEMBL4890265

CCOc1nc(F)cc2nc(S(=O)(=O)Nc3c(Cl)cccc3C(=O)O)nn12.CCOc1nc(F)cc2nc(S(=O)(=O)Nc3c(Cl)cccc3C(=O)O)nn12

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.39
ACLY P53396 2/20 0.35
CCR2 P41597 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CCR4 P51679 1/20 0.35
CCR5 P51681 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL118467 1.00 WDR5 (0.39) WDR5ACLYCCR2CYP1A2CYP3A4
SCHEMBL29396759 1.00 WDR5 (0.39) WDR5ACLYCCR2CYP1A2CYP3A4
SCHEMBL30416435 0.92 CA2 (0.34) WDR5ALDH1A1
SCHEMBL64266 0.92 CA2 (0.34) WDR5ALDH1A1
SCHEMBL22188698 0.91 WDR5 (0.34) WDR5ACLYCCR2CYP1A2CYP3A4
SCHEMBL18643336 0.91 CA2 (0.40) ALDH1A1
Diclosulam SCHEMBL2231960 0.91 CA2 (0.33) WDR5ALDH1A1
SCHEMBL8848603 0.91 WDR5 (0.42) WDR5ALDH1A1
Diclosulam SCHEMBL116344 0.91 GNRHR (0.35) CCR4ALDH1A1SMN1; SMN2
SCHEMBL8848572 0.88 GNRHR (0.34) ACLYCCR4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 135 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3645640-B1 SILICONE-POLYETHER COPOLYMER, METHOD OF PREPARING SAME, AND SEALANT COMPRISING SAME DOW SILICONES CORP (US) 2024-03-06 EP disclosed
WO-2023215360-A1 SILICONE-POLYETHER COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORPORATION (US) 2023-11-09 WO disclosed
US-11807775-B2 Silicone-organic copolymer, sealants comprising same, and related methods DOW SILICONES CORPORATION (US) 2023-11-07 US disclosed
US-11760841-B2 Silicone-polycarbonate copolymer, sealants comprising same, and related methods DOW SILICONES CORPORATION (US) 2023-09-19 US disclosed
EP-3898779-B1 SILICONE-POLYESTER COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORP (US) 2023-02-08 EP disclosed
EP-3898781-B1 SILICONE-POLYCARBONATE COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORP (US) 2023-01-04 EP disclosed
US-20220064383-A1 SILICONE-POLYACRYLATE COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORPORATION 2022-03-03 US disclosed
US-20220064482-A1 SILICONE-ORGANIC COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORPORATION 2022-03-03 US disclosed
EP-3898781-A1 SILICONE-POLYCARBONATE COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS Dow Silicones Corporation (US) 2021-10-27 EP disclosed
EP-3898782-A1 SILICONE-POLYACRYLATE COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS Dow Silicones Corporation (US) 2021-10-27 EP disclosed
WO-2013013111-A1 YTTRIUM CONTAINING COMPLEX AND CONDENSATION REACTION CATALYSTS, METHODS FOR PREPARING THE CATALYSTS, AND COMPOSITIONS CONTAINING THE CATALYSTS DOW CORNING CORPORATION (US) 2013-01-24 WO disclosed
WO-2013012897-A1 COPPER CONTAINING COMPLEX, CONDENSATION REACTION COMPOSITIONS CONTAINING THE COMPLEX, AND METHODS FOR THE PREPARATION AND USE OF THE COMPOSITIONS DOW CORNING CORPORATION (US) 2013-01-24 WO disclosed
WO-2013012977-A1 ZINC CONTAINING COMPLEX AND CONDENSATION REACTION CATALYSTS, METHODS FOR PREPARING THE CATALYSTS, AND COMPOSITIONS CONTAINING THE CATALYSTS DOW CORNING CORPORATION (US) 2013-01-24 WO disclosed
WO-2013013109-A1 GERMANIUM CONTAINING COMPLEX AND CONDENSATION REACTION CURABLE COMPOSITIONS AND METHODS FOR THE PREPARATION AND USE OF THE COMPOSITIONS DOW CORNING CORPORATION (US) 2013-01-24 WO disclosed
WO-2013009836-A1 SAMARIUM CONTAINING COMPLEXES AND CONDENSATION REACTION CATALYSTS, METHODS FOR PREPARING THE CATALYSTS, AND COMPOSITIONS CONTAINING THE CATALYSTS DOW CORNING CORPORATION (US) 2013-01-17 WO disclosed
WO-2013009840-A1 LANTHANIDE COMPLEXES WITH IMIDAZOLE LIGANDS FOR CONDENSATION REACTIONS DOW CORNING CORPORATION (US) 2013-01-17 WO disclosed
WO-2013000788-A1 HYDROSILYLATION REACTION CURABLE COMPOSITIONS AND METHODS FOR THEIR PREPARATION AND USE DOW CORNING CORPORATION (US) 2013-01-03 WO disclosed
US-20080118734-A1 Coating Compositions DOW CORNING IRELAND LTD. (IE) 2008-05-22 US disclosed
EP-1744836-A2 PROCESS AND APPARATUS FOR PLASMA COATING, SUBSTRATES COATED BY THIS METHOD OR APPARATUS Dow Corning Ireland Limited (IE) 2007-01-24 EP disclosed
WO-2005110626-A2 PROCESS AND APPARATUS FOR PLASMA COATING, SUBSTRATES COATED BY THIS METOD OR APPARATUS DOW CORNING IRELAND LIMITED (IE) 2005-11-24 WO disclosed