SCHEMBL4897

SCHEMBL4897

c1csc(-c2ncco2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.49
KDM4E B2RXH2 9/20 0.49
RAB9A P51151 8/20 0.49
NPC1 O15118 7/20 0.49
HPGD P15428 7/20 0.49
SMN1; SMN2 Q16637 6/20 0.49
HSD17B10 Q99714 3/20 0.49
TP53 P04637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GAA P10253 2/20 0.43
LTA4H P09960 1/20 0.43
GFER P55789 1/20 0.43
MAPT P10636 3/20 0.42
POLB P06746 2/20 0.42
CYP2C9 P11712 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoxazole SCHEMBL27894024 0.88 RAB9A (0.41) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL28928822 0.84 SMN1; SMN2 (0.42) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL3220235 0.78 RAB9A (0.39) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL5132723 0.72 ALDH1A1 (0.49) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL13762461 0.70 KDM4E (0.70) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL100765 0.69 HPGDS (0.46) LTA4HHPGDS
SCHEMBL9065298 0.69 HPGDS (0.42) LTA4HCYP1A2CYP2D6CYP3A4HPGDS
SCHEMBL22698306 0.68 LTA4H (0.40) LTA4HMAPTHPGDSHDAC8
SCHEMBL262283 0.68 RAB9A (0.45) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL262142 0.68 KDM4E (0.49) ALDH1A1KDM4ERAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10203 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4337220-A1 SELECTIVE, PARTIAL, AND ARRESTIN-BIASED 5-HT2A AGONISTS WITH UTILITY IN VARIOUS DISORDERS Saint Joseph's University (US) 2024-03-20 EP claimed
CN-116003433-A Organic photosensitive molecule with spectral response reaching infrared region and application thereof 广州光达创新科技有限公司 2023-04-25 CN claimed
US-20220396571-A1 SPIROPIPERIDINE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS MERCK SHARP & DOHME CORP. (US) 2022-12-15 US claimed
CN-114891027-A Infrared-response N-type organic molecule and application thereof 广州光达创新科技有限公司 2022-08-12 CN claimed
CN-113683616-A KRAS G12C mutein inhibitors 广州百霆医药科技有限公司 2021-11-23 CN claimed
CN-113527300-A Bruton's tyrosine protein kinase inhibitor 广州百霆医药科技有限公司 2021-10-22 CN claimed
EP-3253764-B1 MACROCYCLIC COMPOUNDS AS IRAK1/4 INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2021-06-09 EP claimed
US-10870630-B2 Substituted bicyclic heteroaryl allosteric modulators of nicotinic acetylcholine receptors MERCK SHARP & DOHME CORP. 2020-12-22 US claimed
EP-3253763-B1 PYRIDAZINONE MACROCYCLES AS IRAK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2020-09-30 EP claimed
US-20200246274-A1 GLUTAMINASE INHIBITOR DISCOVERY AND NANOPARTICLE-ENHANCED DELIVERY FOR CANCER THERAPY THE JOHNS HOPKINS UNIVERSITY 2020-08-06 US claimed
US-6124302-A TREATING HIV INFECTIONS DUPONT PHARMACEUTICALS (US) 2000-09-26 US claimed
WO-2000047553-A2 ALKENYL AND ALKYNYL COMPOUNDS AS INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC. (US) 2000-08-17 WO claimed
CN-1261345-A Glyoxylic acid amides BAYER AG (DE) 2000-07-26 CN claimed
CN-1216043-A Substd. benzenesulfonamide derivs as prodrugs of COX-2 inhibitors SEARLE & CO (US) 1999-05-05 CN claimed
CN-1095591-A The associating of a kind of cholesteral biosynthesis inhibitor and a kind of beta-lactam cholesterol absorption inhibitor SCHERING CORP (US) 1994-11-30 CN claimed
CN-1069024-A As 'beta '-lactam compounds that reduces the replacement of cholesterol medicament in the blood and preparation method thereof SCHERING CORP (US) 1993-02-17 CN claimed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP claimed
US-4980348-A HETEROANELLATED PHENYLGLYCINE-BETA-LACTAM ANTIBIOTICS BAYER AKTIENGESELLSCHAFT (DE) 1990-12-25 US claimed
CN-88103202-A Vinyl cephalosporin compound that replaces and preparation method thereof and as the application of medicine 1988-12-21 CN claimed
US-4147789-A ANTIPARKINSON AGENTS SANDOZ LTD. (CH) 1979-04-03 US claimed