SCHEMBL4903029

SCHEMBL4903029

COC(=O)c1cc(S(=O)(=O)NCCOc2cc(Cl)cc(Cl)c2)ccc1C

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
HTT P42858 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
NPSR1 Q6W5P4 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
GAA P10253 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 1/20 0.45
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4899741 0.91 LMNA (0.56) TDP1HTTMEN1KMT2ANPSR1
SCHEMBL4906713 0.82 TDP1 (0.59) TDP1HTTMEN1KMT2ANPSR1
SCHEMBL4902606 0.82 TDP1 (0.51) TDP1HTTMEN1KMT2ANPSR1
SCHEMBL4909535 0.81 TDP1 (0.57) TDP1HTTMEN1KMT2ANPSR1
SCHEMBL4905142 0.79 MAPT (0.50) HTTMEN1KMT2ANPSR1GAA
SCHEMBL4907392 0.78 TDP1 (0.47) TDP1HTTMEN1KMT2ANPSR1
SCHEMBL4900651 0.78 LMNA (0.52) HTTKMT2ASMN1; SMN2LMNAALDH1A1
SCHEMBL4895834 0.77 MAPT (0.56) MEN1KMT2ANPSR1SMN1; SMN2LMNA
SCHEMBL4906669 0.77 ALDH1A1 (0.60) HTTMEN1KMT2ANPSR1GAA
SCHEMBL4895764 0.77 MAPT (0.54) MEN1KMT2ANPSR1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20050288340-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER INC 2005-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288340-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PPARA, PPARG, PPARD TDP1 3653/4885HTT 696/4885MEN1 4855/4885
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PPARA, PPARG, PPARD TDP1 3653/4885HTT 696/4885MEN1 4855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.