SCHEMBL4904141

SCHEMBL4904141

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C)CC3)nc21

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.79
CYP2C9 P11712 1/20 0.79
ATP6V1B2 P21281 1/20 0.79
TBXA2R P21731 1/20 0.79
EDNRA P25101 1/20 0.79
TARBP2 Q15633 1/20 0.79
DRD3 P35462 1/20 0.64
KDM4E B2RXH2 8/20 0.59
ALDH1A1 P00352 4/20 0.59
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
HPGD P15428 2/20 0.59
NPC1 O15118 1/20 0.59
CASP1 P29466 1/20 0.53
ABCC4 O15439 1/20 0.51
PKM P14618 1/20 0.51
PTGS1 P23219 1/20 0.51
HSD17B10 Q99714 2/20 0.51
GAA P10253 1/20 0.51
RAD52 P43351 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11007797 0.92 LMNA (0.67) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL8044673 0.92 LMNA (0.79) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL11153426 0.91 LMNA (0.82) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL10028900 0.90 LMNA (0.81) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL10108591 0.89 LMNA (0.75) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL12665451 0.89 LMNA (0.75) LMNACYP2C9ATP6V1B2TBXA2REDNRA
Enoxacin SCHEMBL29384458 0.88 LMNA (1.00) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL11080390 0.88 LMNA (0.78) LMNACYP2C9ATP6V1B2TBXA2REDNRA
Enoxacin SCHEMBL33963 0.88 LMNA (1.00) LMNACYP2C9ATP6V1B2TBXA2REDNRA
Enoxacin SCHEMBL2635855 0.88 LMNA (1.00) LMNACYP2C9ATP6V1B2TBXA2REDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112824405-B Acrylic ketone derivative of N-methyl enoxacin and preparation method and application thereof 河南大学 2023-06-02 CN disclosed
US-8231897-B2 Hydrostatic delivery system for controlled delivery of agent MACGREGOR ALEXANDER (CA) 2012-07-31 US disclosed
US-20080317847-A1 HYDROSTATIC DELIVERY SYSTEM FOR CONTROLLED DELIVERY OF AGENT MACGREGOR ALEXANDER 2008-12-25 US disclosed
US-7381424-B2 Hydrostatic delivery system for controlled delivery of agent MACGREGOR ALEXANDER 2008-06-03 US disclosed
EP-1347748-A2 HYDROSTATIC DELIVERY SYSTEM FOR CONTROLLED DELIVERY OF AGENT MacGregor, Alexander (CA) 2003-10-01 EP disclosed
US-20020155067-A1 Hydrostatic delivery system for controlled delivery of agent MACGREGOR ALEXANDER (CA) 2002-10-24 US disclosed
WO-2002045695-A2 HYDROSTATIC DELIVERY SYSTEM FOR CONTROLLED DELIVERY OF AGENT MACGREGOR ALEXANDER (CA) 2002-06-13 WO disclosed
EP-0169105-B1 CONTROLLED POROSITY OSMOTIC PUMP MERCK & CO. INC. (US) 1991-08-07 EP disclosed
US-4968507-A SUSTAINED RELEASE OF DRUG MERCK & CO., INC. (US) 1990-11-06 US disclosed
EP-0208617-B1 CONTROLLED DRUG DEVICE AND PROCESS FOR CATALYSING THE EROSION OF AN ACID LABILE POLYMER MERCK & CO. INC. (US) 1990-09-26 EP disclosed
US-4851228-A Multiparticulate controlled porosity osmotic MERCK & CO., INC. (US) 1989-07-25 US disclosed
US-4780319-A DRUG DELIVERY USING POLYORTHOESTERS COATINGS MERCK & CO., INC. (US) 1988-10-25 US disclosed
EP-0208617-A1 Controlled drug device and process for catalysing the erosion of an acid labile polymer MERCK & CO. INC. (US) 1987-01-14 EP disclosed
EP-0169105-A2 Controlled porosity osmotic pump MERCK & CO. INC. (US) 1986-01-22 EP disclosed
US-4496566-A ANTIBACTERIAL AGENT DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1985-01-29 US disclosed
US-4359578-A Naphthyridine derivatives and salts thereof useful as antibacterial agents DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1982-11-16 US disclosed
US-4352803-A BACTERICIDES DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1982-10-05 US disclosed
EP-0009425-A1 Novel naphtyridine derivatives and pharmaceutical compositions containing them Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1980-04-02 EP disclosed