SCHEMBL4907955

SCHEMBL4907955

CCOC(=O)c1cnc(C)c(-n2cc(C(=O)NCC(C)(C)C)nn2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 1/20 0.38
ACKR3 P25106 2/20 0.35
DDT P30046 2/20 0.35
KMT2A Q03164 1/20 0.35
MIF P14174 1/20 0.35
SPR P35270 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA12 O43570 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CNR2 P34972 1/20 0.34
P2RY12 Q9H244 2/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781668 0.88 MIF (0.39) ACKR3DDTMIFCYP2C9CNR2
SCHEMBL14293530 0.83 ESRRA (0.40) ESRRASPRCYP2C9CYP2C19CA1
SCHEMBL4782960 0.83 CYP2C19 (0.46) ESRRASPRCYP2C9CYP2C19CA1
SCHEMBL14292741 0.82 MIF (0.38) ESRRAACKR3DDTMIFCNR2
SCHEMBL4780603 0.79 DRD2 (0.38) ACKR3DDTMIFCYP2C19CNR2
SCHEMBL4782176 0.79 BRAF (0.45) LMNAMAPT
SCHEMBL4784135 0.77 CYP1A2 (0.48) KMT2ACYP2C9CYP2C19
SCHEMBL4782660 0.76 NR1I2 (0.42) DDTMIF
SCHEMBL4782271 0.76 MAPK14 (0.39) DDTCYP2C9CYP2C19
SCHEMBL4781910 0.75 GSK3A (0.33) DDTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed