SCHEMBL4782960

SCHEMBL4782960

CCOC(=O)c1cnc(C)c(-n2cc(C(=O)O)nn2)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 1/20 0.46
ESRRA P11474 1/20 0.42
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
PFKFB3 Q16875 1/20 0.38
SPR P35270 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14293530 0.86 ESRRA (0.40) CYP2C19CYP2C9ESRRAALDH1A1LMNA
SCHEMBL4907955 0.83 ESRRA (0.38) CYP2C19CYP2C9ESRRAALDH1A1LMNA
SCHEMBL13436160 0.77 LMNA (0.38) CYP2C19CYP2C9ESRRAALDH1A1LMNA
SCHEMBL1404531 0.75 ALDH1A1 (0.48) CYP2C19CYP2C9ESRRAALDH1A1LMNA
SCHEMBL4782153 0.73 NOTUM (0.37) ALDH1A1SMN1; SMN2
SCHEMBL4782157 0.73 NOTUM (0.37) ALDH1A1SMN1; SMN2
SCHEMBL5481626 0.72 CYP2C9 (0.59) CYP2C19CYP2C9ALDH1A1LMNACA1
SCHEMBL3120898 0.71 TSHR (0.50) LMNA
SCHEMBL26412819 0.70 CYP2C9 (0.56) CYP2C19CYP2C9LMNACA1CA2
SCHEMBL14293383 0.70 RXRA (0.35) ESRRACA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed