SCHEMBL4911020

SCHEMBL4911020

O=C(CNc1ccc(Cl)cc1F)Nc1ccccc1C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.62
KMT2A Q03164 4/20 0.62
NPSR1 Q6W5P4 3/20 0.62
MAPT P10636 3/20 0.62
MEN1 O00255 3/20 0.62
LMNA P02545 1/20 0.62
TDP1 Q9NUW8 1/20 0.57
GRIK1 P39086 2/20 0.53
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
HPGD P15428 1/20 0.50
KDM4E B2RXH2 4/20 0.48
GAA P10253 2/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
ATM Q13315 1/20 0.48
HCAR2 Q8TDS4 1/20 0.48
POLB P06746 1/20 0.47
G6PD P11413 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689589 0.90 ALDH1A1 (0.64) ALDH1A1KMT2ANPSR1MAPTMEN1
SCHEMBL8693363 0.88 GRIK1 (0.70) ALDH1A1KMT2ANPSR1MAPTMEN1
SCHEMBL8689403 0.85 ALDH1A1 (0.59) ALDH1A1KMT2AMAPTMEN1LMNA
SCHEMBL4906943 0.85 LMNA (0.55) ALDH1A1KMT2ANPSR1MAPTMEN1
SCHEMBL4912702 0.85 RAB9A (0.59) ALDH1A1KMT2ANPSR1MAPTMEN1
SCHEMBL4650557 0.84 KDM4E (0.53) ALDH1A1KMT2ANPSR1MAPTMEN1
SCHEMBL4650555 0.83 KDM4E (0.59) ALDH1A1KMT2ANPSR1MAPTMEN1
SCHEMBL4913029 0.81 KDM4E (0.68) ALDH1A1KMT2AMAPTMEN1RAB9A
SCHEMBL8478866 0.80 HDAC1 (0.55) ALDH1A1KMT2AMAPTMEN1LMNA
SCHEMBL8482273 0.80 KMT2A (0.55) ALDH1A1KMT2AMAPTMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2008-10-30 US claimed
US-7408078-B2 Anthranilic acid derivatives useful in treating infection with hepatitis C virus WYETH (US) 2008-08-05 US claimed
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus VIROPHARMA INCORPORATED 2005-01-06 US claimed
WO-2004091724-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2004-10-28 WO claimed
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2008-10-30 US disclosed
US-7408078-B2 Anthranilic acid derivatives useful in treating infection with hepatitis C virus WYETH (US) 2008-08-05 US disclosed
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus VIROPHARMA INCORPORATED 2005-01-06 US disclosed
WO-2004091724-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2004-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus HCCS, ALAD, HAVCR2 ALDH1A1 271/4885KMT2A 1394/4885NPSR1 1784/4885
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS HCCS, ALAD, HAVCR2 ALDH1A1 271/4885KMT2A 1394/4885NPSR1 1784/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.