SCHEMBL4911501

SCHEMBL4911501

COc1cc(I)c(C(=O)N(c2cnnc3ccc([N+](=O)[O-])cc23)C(C)N(C)C)cc1OC

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
MAPT P10636 2/20 0.36
AMY1A P0DUB6 2/20 0.35
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
LMNA P02545 3/20 0.33
KDM4E B2RXH2 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
POLB P06746 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
KCNMA1 Q12791 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4911505 0.83 ALDH1A1 (0.40) ALDH1A1MAPTAMY1AHTTKDM4E
Dimethylamine SCHEMBL4911507 0.81 ALDH1A1 (0.40) ALDH1A1MAPTAMY1AHTTLMNA
SCHEMBL4903308 0.73 ALDH1A1 (0.39) ALDH1A1MAPTAMY1AHTTSMN1; SMN2
SCHEMBL241748 0.70 KMT2A (0.36) ALDH1A1HTTLMNAKDM4EKMT2A
SCHEMBL240953 0.69 ALDH1A1 (0.33) ALDH1A1HTTSMN1; SMN2LMNAKDM4E
SCHEMBL4910912 0.68 MAPT (0.38) ALDH1A1MAPTAMY1ASMN1; SMN2LMNA
SCHEMBL13996173 0.65 ALDH1A1 (0.36) ALDH1A1MAPTHTTLMNAKDM4E
SCHEMBL4903280 0.61 TXNRD1 (0.47) ALDH1A1SMN1; SMN2ABCG2
SCHEMBL17478755 0.60 ALDH1A1 (0.71) ALDH1A1MAPTAMY1AHTTKMT2A
SCHEMBL5779054 0.60 L3MBTL1 (0.48) ALDH1A1MAPTHTTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080045538-A1 Nitro and amino substituted topoisomerase agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2008-02-21 US disclosed
US-6992089-B2 Nitro and amino substituted topoisomerase agents RUTGERS, THE UNIVERSITY OF NEW JERSEY (US) 2006-01-31 US disclosed
US-20040102443-A1 Nitro and amino substituted topoisomerase agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2004-05-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045538-A1 Nitro and amino substituted topoisomerase agents TOP1, TOP2A, TOP2B ALDH1A1 2380/4885MAPT 4024/4885AMY1A 3370/4885
US-20040102443-A1 Nitro and amino substituted topoisomerase agents TOP1, TOP2A, TOP2B ALDH1A1 1476/4885MAPT 4283/4885AMY1A 2151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.