Fumaric Acid

Fumaric Acid

SCHEMBL4916656

CCC[N+](C)(CCC)CCC.CCC[N+](C)(CCC)CCC.O=C([O-])/C=C/C(=O)[O-]

nearest known ligand 0.48

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Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BBOX1 O75936 6/20 0.46
FFAR3 O14843 2/20 0.35
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
CA1 P00915 2/20 0.33
CA9 Q16790 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
CYP3A4 P08684 2/20 0.31
TSHR P16473 2/20 0.31
NFKB1 P19838 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL4917899 1.00 BBOX1 (0.46) BBOX1FFAR3HDAC3HDAC1HDAC2
Fumaric Acid SCHEMBL4951203 1.00 BBOX1 (0.46) BBOX1FFAR3HDAC3HDAC1HDAC2
Fumaric Acid SCHEMBL4929332 0.98 BBOX1 (0.45) BBOX1FFAR3HDAC3HDAC1HDAC2
Fumaric Acid SCHEMBL4929679 0.98 BBOX1 (0.45) BBOX1FFAR3HDAC3HDAC1HDAC2
Fumaric Acid SCHEMBL4929346 0.98 BBOX1 (0.45) BBOX1FFAR3HDAC3HDAC1HDAC2
Fumaric Acid SCHEMBL4925561 0.92 BBOX1 (0.41) BBOX1TSHR
Fumaric Acid SCHEMBL4953243 0.92 BBOX1 (0.41) BBOX1TSHR
Fumaric Acid SCHEMBL4924908 0.92 BBOX1 (0.41) BBOX1TSHR
Tributylmethylammonium SCHEMBL4952826 0.86 BBOX1 (0.45) BBOX1CA1CES2CES1
Tributylmethylammonium SCHEMBL4931562 0.86 BBOX1 (0.45) BBOX1CA1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080312351-A1 Tetraalkylammonium Carboxylate Salts as Trimerization Catalysts for Spray Foam Applications AIR PRODUCTS AND CHEMICALS, INC. (US) 2008-12-18 US claimed
EP-2003157-A2 Tetraalkylammonium carboxylate salts as trimerization catalysts for spray foam applications Air Products and Chemicals, Inc. (US) 2008-12-17 EP claimed
US-20080312351-A1 Tetraalkylammonium Carboxylate Salts as Trimerization Catalysts for Spray Foam Applications AIR PRODUCTS AND CHEMICALS, INC. (US) 2008-12-18 US disclosed
EP-2003157-A2 Tetraalkylammonium carboxylate salts as trimerization catalysts for spray foam applications Air Products and Chemicals, Inc. (US) 2008-12-17 EP disclosed