Tofenacin

Tofenacin

SCHEMBL49290

CNCCOC(c1ccccc1)c1ccccc1C

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.64
SLC6A2 P23975 5/20 0.64
HTR2A P28223 5/20 0.64
HRH1 P35367 5/20 0.64
CYP3A4 P08684 4/20 0.64
CHRM1 P11229 4/20 0.64
ADRA2B P18089 4/20 0.64
HTR2C P28335 4/20 0.64
SLC6A4 P31645 4/20 0.64
OPRM1 P35372 4/20 0.64
DRD3 P35462 4/20 0.64
HTR2B P41595 4/20 0.64
SLC6A3 Q01959 4/20 0.64
KCNH2 Q12809 4/20 0.64
CHRM2 P08172 2/20 0.64
CHRM4 P08173 2/20 0.64
CHRM5 P08912 2/20 0.64
ADRA2A P08913 2/20 0.64
CHRM3 P20309 2/20 0.64
HRH2 P25021 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tofenacin SCHEMBL637494 0.98 LMNA (0.65) CYP2D6SLC6A2HTR2AHRH1CYP3A4
SCHEMBL4667597 0.87 CYP2D6 (0.76) CYP2D6SLC6A2HTR2AHRH1CYP3A4
SCHEMBL3333230 0.85 SIGMAR1 (0.68) CYP2D6SLC6A2HTR2AHRH1CHRM1
Hydrochloric Acid SCHEMBL28100967 0.83 HTT (0.69) CYP2D6SLC6A2HTR2AHRH1CHRM1
SCHEMBL25375446 0.81 CYP2D6 (0.68) CYP2D6SLC6A2HTR2AHRH1CYP3A4
SCHEMBL4669319 0.81 CYP2D6 (0.68) CYP2D6SLC6A2HTR2AHRH1CYP3A4
SCHEMBL8105789 0.78 CYP2D6 (0.64) CYP2D6SLC6A2HTR2AHRH1CYP3A4
Orphenadrine SCHEMBL119471 0.78 SLC6A2 (1.00) CYP2D6SLC6A2HTR2AHRH1CYP3A4
Orphenadrine SCHEMBL28727 0.78 SLC6A2 (1.00) CYP2D6SLC6A2HTR2AHRH1CYP3A4
Orphenadrine SCHEMBL29359844 0.78 SLC6A2 (1.00) CYP2D6SLC6A2HTR2AHRH1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2359 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12496300-B2 Methods of treating acute depression and anxiety INTRA-CELLULAR THERAPIES, INC. (US) 2025-12-16 US claimed
EP-4479032-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS Sage Therapeutics, Inc. (US) 2024-12-25 EP claimed
CN-119072304-A Neuroactive steroids for the treatment of CNS related disorders 萨奇治疗股份有限公司 2024-12-03 CN claimed
EP-3706762-B1 N4-HYDROXYCYTIDINE DERIVATIVE AND ANTI-VIRAL USES RELATED THERETO UNIV EMORY (US) 2024-10-16 EP claimed
US-20240307386-A1 NOVEL METHODS INTRA-CELLULAR THERAPIES, INC. 2024-09-19 US claimed
WO-2023159035-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS SAGE THERAPEUTICS, INC. (US) 2023-08-24 WO claimed
WO-2023158668-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS SAGE THERAPEUTICS, INC. (US) 2023-08-24 WO claimed
CN-114869838-A Soothing and moisturizing composition and preparation method and application thereof 广州市科能化妆品科研有限公司 2022-08-09 CN claimed
WO-2022159506-A1 DEUTERATED CANNABIDIOL COMPOUNDS MERIT THERAPEUTICS, INC. (US) 2022-07-28 WO claimed
WO-2022159507-A1 COMBINATION OF CANNABINOIDS WITH ADDITIONAL THERAPEUTIC AGENTS FOR TREATING DISEASES OR DISORDERS MERIT THERAPEUTICS, INC. (US) 2022-07-28 WO claimed
US-20020161016-A1 As-needed administration of tricyclic and other non-SRI antidepressant drugs to treat premature ejaculation VIVUS LLC (F/K/A VIVUS, INC.) 2002-10-31 US claimed
WO-2002080708-A2 A SMOKER'S REQUISITE ENSLIN GEORGE FREDERICK (ZA) 2002-10-17 WO claimed
US-6403597-B1 PRETREATMENT SEXUAL INTERCOURSE VIVUS, INC. 2002-06-11 US claimed
WO-2002041883-A2 AS-NEEDED ADMINISTRATION OF TRICYCLIC AND OTHER NON-SRI ANTIDEPRESSANT DRUGS TO TREAT PREMATURE EJACULATION VIVUS, INC. (US) 2002-05-30 WO claimed
US-20020037828-A1 Administration of phosphodiesterase inhibitors for the treatment of premature ejaculation VIVUS, INC. 2002-03-28 US claimed
US-20010008896-A1 Administration of active agents, including 5-HT receptor agonists and antagonists, to treat premature ejaculation SMITH WILLIAM L (US) 2001-07-19 US claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5922341-A Local administration of pharmacologically active agents to treat premature ejaculation VIVUS, INCORPORATED (US) 1999-07-13 US claimed