SCHEMBL492906

SCHEMBL492906

Cc1cc(C)c(S(=O)(=O)N2CCC(OCC(=O)NC3CCC(C(c4ccccc4)N(C)C)CC3)C2)c(C)c1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 17/20 0.47
EBP Q15125 1/20 0.42
DHCR7 Q9UBM7 1/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493328 0.93 BDKRB1 (0.41) EPHX2EBPDHCR7MEN1KMT2A
SCHEMBL493537 0.92 EPHX2 (0.41) EPHX2EBPDHCR7MEN1KMT2A
SCHEMBL493908 0.92 EPHX2 (0.41) EPHX2EBPDHCR7
SCHEMBL493296 0.89 EPHX2 (0.48) EPHX2EBPDHCR7MEN1KMT2A
SCHEMBL493571 0.89 KMT2A (0.46) EPHX2MEN1KMT2A
SCHEMBL492633 0.88 KMT2A (0.45) EPHX2MEN1KMT2A
SCHEMBL493757 0.88 KMT2A (0.39) EPHX2MEN1KMT2A
SCHEMBL492404 0.88 EPHX2 (0.40) EPHX2EBPDHCR7
SCHEMBL492916 0.86 BDKRB1 (0.40) EPHX2MEN1KMT2A
SCHEMBL493194 0.85 BDKRB1 (0.39) EPHX2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106055-B2 Substituted amide compounds GRUENENTHAL GMBH (DE) 2012-01-31 US claimed
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP claimed
US-20080306084-A1 Substituted Amide Compounds GRUENENTHAL GMBH (DE) 2008-12-11 US claimed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO claimed
US-8106055-B2 Substituted amide compounds GRUENENTHAL GMBH (DE) 2012-01-31 US disclosed
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP disclosed
US-20080306084-A1 Substituted Amide Compounds GRUENENTHAL GMBH (DE) 2008-12-11 US disclosed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306084-A1 Substituted Amide Compounds OPRK1, NAA50, ACMSD EPHX2 2567/4885EBP 293/4885DHCR7 3298/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.