SCHEMBL4930261

SCHEMBL4930261

Cc1ccc(-c2cccc(F)c2OCCN2CCCC2)cc1N1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.47
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.40
HTR6 P50406 3/20 0.39
SRC P12931 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
HTR1A P08908 2/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5577195 0.84 HTR7 (0.43) HTR7HTR6HTR1A
SCHEMBL4933067 0.84 HTR7 (0.54) HTR7ALDH1A1TDP1ESR1ESR2
SCHEMBL4932567 0.81 ALDH1A1 (0.46) ALDH1A1POLBSRCTDP1ESR1
SCHEMBL1790594 0.79 RPS6KB1 (0.41)
Trifluoroacetic Acid SCHEMBL4931987 0.78 KDM4E (0.52) HTR7ALDH1A1POLBTDP1
SCHEMBL4930427 0.77 KDM4E (0.48) ALDH1A1POLBSRCHTR1A
SCHEMBL11357385 0.68 ALDH1A1 (0.62) HTR7ALDH1A1POLBTDP1
Hydrochloric Acid SCHEMBL4928899 0.67 HTR6 (0.61) HTR7ALDH1A1HTR6HTR1A
SCHEMBL21555229 0.67 TSHR (0.50) ALDH1A1POLBTDP1
SCHEMBL14559927 0.66 HTR1A (0.59) HTR6TDP1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8076338-B2 Such as 6-(4-phenylpiperazin-1-yl)-9H-purine; cell proliferation/differentiation EXELIXIS, INC. (US) 2011-12-13 US disclosed
US-20080076774-A1 Kinase Modulators and Methods of Use EXELIXIS, INC. (US) 2008-03-27 US disclosed
EP-1750727-A2 KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2007-02-14 EP disclosed
WO-2005117909-A2 KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2005-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080076774-A1 Kinase Modulators and Methods of Use AKT3, RPS6KA3, CDK3 HTR7 2882/4885ALDH1A1 4305/4885POLB 2210/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.