SCHEMBL4938426

SCHEMBL4938426

Cc1ccc(C(=O)CCC(C)C)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.60
TRPA1 O75762 1/20 0.56
GSK3B P49841 1/20 0.53
CTNNB1 P35222 3/20 0.50
WNT3A P56704 3/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474694 0.84 HSD17B3 (0.62) TRPA1NPC1RAB9AALDH1A1USP5
SCHEMBL16552778 0.83 KMT2A (0.83) KMT2AGSK3BCTNNB1WNT3ANPC1
SCHEMBL17032601 0.82 NPC1 (0.62) KMT2ATRPA1CTNNB1NPC1RAB9A
SCHEMBL7426211 0.82 TRPA1 (0.54) KMT2ATRPA1GSK3BNPC1RAB9A
SCHEMBL2850064 0.82 TRPA1 (0.54) KMT2ATRPA1GSK3BMEN1ALDH1A1
SCHEMBL725762 0.82 TRPA1 (0.58) KMT2ATRPA1GSK3BCTNNB1WNT3A
Benzene SCHEMBL27311002 0.82 TRPA1 (0.58) KMT2ATRPA1GSK3BCTNNB1WNT3A
SCHEMBL9441163 0.81 TRPA1 (0.53) KMT2ATRPA1MEN1ALDH1A1LMNA
SCHEMBL15656585 0.81 TRPA1 (0.53) KMT2ATRPA1NPC1RAB9AMEN1
SCHEMBL13220674 0.79 SMN1; SMN2 (0.66) TRPA1GSK3BNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2735581-B1 COMPOSITION AND POLYMER ASAHI CHEMICAL IND (JP) 2021-07-14 EP disclosed
US-9738757-B2 Composition and polymer ASAHI KASEI CHEMICALS CORPORATION (JP) 2017-08-22 US disclosed
US-20160222168-A1 Composition and Polymer ASAHI KASEI CHEMICALS CORPORATION (JP) 2016-08-04 US disclosed
US-9334371-B2 Composition and polymer ASAHI KASEI CHEMICALS CORPORATION (JP) 2016-05-10 US disclosed
EP-2735581-A1 COMPOSITION AND POLYMER Asahi Kasei Chemicals Corporation (JP) 2014-05-28 EP disclosed
US-20140121293-A1 Composition and Polymer ASAHI KASEI CHEMICALS CORPORATION (JP) 2014-05-01 US disclosed
US-20080234498-A1 Pyrovalerone Analogues and Therapeutic Uses Thereof PRESIDENT AND FELLOW OF HARVARD COLLEGE (US) 2008-09-25 US disclosed
EP-1670755-A4 PYROVALERONE ANALOGS AND THERAPEUTIC USES THEREOF HARVARD COLLEGE (US) 2007-02-28 EP disclosed
EP-1670755-A2 PYROVALERONE ANALOGS AND THERAPEUTIC USES THEREOF President And Fellows of Harvard College (US) 2006-06-21 EP disclosed
WO-2005034878-A2 PYROVALERONE ANALOGS AND THERAPEUTIC USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2005-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234498-A1 Pyrovalerone Analogues and Therapeutic Uses Thereof SLC6A2, SLC6A4, SLC6A3 KMT2A 3331/4885TRPA1 722/4885GSK3B 539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.