SCHEMBL4940341

SCHEMBL4940341

CS(=O)(=O)c1ccc(-c2ccsc2)c(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.51
ACMSD Q8TDX5 1/20 0.46
IDH2 P48735 10/20 0.43
EIF4E P06730 1/20 0.42
PTGS2 P35354 2/20 0.41
GPR35 Q9HC97 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4934685 0.85 NR4A2 (0.44) IDH2PTGS2
SCHEMBL13893700 0.82 PTGS2 (0.44) IDH2PTGS2
SCHEMBL3875822 0.80 LMNA (0.58) LMNAPTGS2
SCHEMBL3873005 0.79 LMNA (0.54) LMNAEIF4EPTGS2
SCHEMBL15025193 0.78 ACMSD (0.59) ACMSDEIF4EGPR35
SCHEMBL12506050 0.78 PTGS2 (0.46) IDH2PTGS2
SCHEMBL12050154 0.77 ACMSD (0.51) ACMSDEIF4EGPR35
SCHEMBL1812902 0.77 PTGS2 (0.58) LMNAPTGS2
SCHEMBL8259316 0.77 LMNA (0.54) LMNAPTGS2
SCHEMBL3875280 0.77 LMNA (0.62) LMNAEIF4EPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080255144-A1 Acylated Piperidines as Glycine Transporter Inhibitors GLAXO GROUP LIMITED 2008-10-16 US disclosed
US-20080255144-A1 Acylated Piperidines as Glycine Transporter Inhibitors GLAXO GROUP LIMITED 2008-10-16 US disclosed
US-20080255144-A1 Acylated Piperidines as Glycine Transporter Inhibitors GLAXO GROUP LIMITED 2008-10-16 US disclosed
EP-1858869-A1 ACYLATED PIPERIDINES AS GLYCINE TRANSPORTER INHIBITORS GLAXO GROUP LIMITED (GB) 2007-11-28 EP disclosed
WO-2006094842-A1 ACYLATED PIPERIDIHES AS GLYCINE TRANSPORTER INHIBITORS GLAXO GROUP LIMITED (GB) 2006-09-14 WO disclosed
WO-2006094842-A1 ACYLATED PIPERIDIHES AS GLYCINE TRANSPORTER INHIBITORS GLAXO GROUP LIMITED (GB) 2006-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080255144-A1 Acylated Piperidines as Glycine Transporter Inhibitors SLC1A1, SLC6A7, SLC1A2 LMNA 4248/4885ACMSD 2234/4885IDH2 1694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.