SCHEMBL4940862

SCHEMBL4940862

Bc1ccc2c(C(N)=O)n(-c3ccc(F)cc3)nc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.44
AURKA O14965 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CDK8 P49336 1/20 0.44
NEK2 P51955 1/20 0.44
LIMK1 P53667 1/20 0.44
CDK5 Q00535 1/20 0.44
DYRK1A Q13627 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
CCNA2 P20248 2/20 0.39
CDK2 P24941 2/20 0.39
CCNA1 P78396 2/20 0.39
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA9 Q16790 1/20 0.36
SCN9A Q15858 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9108907 0.84 CDK5 (0.44) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL4940858 0.76 ESR2 (0.44) MEN1KMT2ALMNAPTGS1PTGS2
SCHEMBL2721702 0.72 CHEK1 (0.54) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL9910900 0.70 CHEK1 (0.59) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL9107560 0.68 SLC2A1 (0.46) NPC1RAB9A
SCHEMBL29161027 0.68 CHEK1 (0.56) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL2721640 0.67 PTGS2 (0.46) PTGS2
SCHEMBL15940565 0.67 CHEK1 (0.51) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL4942119 0.66 CHEK1 (0.46) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL15940529 0.64 NPC1 (0.42) MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012051659-A1 VIRAL POLYMERASE INHIBITORS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2012-04-26 WO disclosed