SCHEMBL4947992

SCHEMBL4947992

COc1cc(-c2cccc(C3=NC(C(F)(F)F)=CCC3=O)c2)cc([N+](=O)[O-])c1O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ABCB1 P08183 6/20 0.38
ABCC1 P33527 6/20 0.38
ERN1 O75460 1/20 0.37
CSNK2A2 P19784 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
GRK6 P43250 1/20 0.35
MAPT P10636 1/20 0.35
TTR P02766 1/20 0.35
LMNA P02545 1/20 0.35
SIRT1 Q96EB6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4950976 0.88 CRHBP (0.42) MEN1ALDH1A1KMT2AABCC1ERN1
SCHEMBL4948139 0.82 FYN (0.40) MEN1KMT2AMAPTLMNA
SCHEMBL3579413 0.75 SMN1; SMN2 (0.42) ALOX5MEN1ALDH1A1KMT2AABCB1
SCHEMBL1446971 0.72 ABCC1 (0.40) ALOX5MEN1ALDH1A1KMT2AL3MBTL1
SCHEMBL4948557 0.62 TTR (0.51) MEN1ALDH1A1KMT2AL3MBTL1ABCB1
SCHEMBL7367724 0.61 TTR (0.57) MEN1ALDH1A1KMT2AABCB1ABCC1
SCHEMBL12118500 0.61 GPR35 (0.57) MEN1ALDH1A1KMT2AERN1MAPT
SCHEMBL3590761 0.61 CRHBP (0.49) ABCC1ERN1CRHBPCRHR2MAPT
SCHEMBL3584563 0.61 TTR (0.53) MEN1ALDH1A1KMT2AL3MBTL1ABCB1
SCHEMBL20022338 0.61 TTR (0.66) MEN1ALDH1A1KMT2AL3MBTL1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed