SCHEMBL4949929

SCHEMBL4949929

O=CN1CCCC1c1cc2ccccc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.41
HRH3 Q9Y5N1 4/20 0.40
AKR1C3 P42330 4/20 0.38
HTR7 P34969 1/20 0.36
ADRA1B P35368 1/20 0.36
MAOB P27338 1/20 0.36
CHRNA7 P36544 1/20 0.36
HRH4 Q9H3N8 1/20 0.35
FAAH O00519 1/20 0.35
SLC6A3 Q01959 3/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985432 0.82 HRH3 (0.39) HRH3AKR1C3CHRNA7HRH4FAAH
SCHEMBL13634946 0.78 CHRNB2 (0.50) HRH3CHRNA7
SCHEMBL13162089 0.78 HRH3 (0.42) HRH3AKR1C3HTR7ADRA1BCHRNA7
SCHEMBL12993141 0.75 CYP2A6 (0.44) CYP2A6HRH3AKR1C3HTR7ADRA1B
SCHEMBL3260435 0.74 CYP2A6 (0.37) CYP2A6AKR1C3MAOBHRH4SLC6A3
SCHEMBL9463940 0.72 HRH3 (0.43) HRH3AKR1C3CHRNA7
SCHEMBL13330544 0.71 CHRNB2 (0.55) CHRNA7
SCHEMBL16343091 0.70 DRD2 (0.54) HRH3AKR1C3
SCHEMBL28152135 0.70 PARP1 (0.50) HRH3AKR1C3CHRNA7HRH4SLC6A4
Hydrochloric Acid SCHEMBL28334700 0.69 PARP1 (0.49) HRH3AKR1C3CHRNA7HRH4SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912976-B1 INDOL-3-YL-CARBONYL-PIPERIDIN-BENZOIMIDAZOLE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2008-11-12 EP disclosed