SCHEMBL4955338

SCHEMBL4955338

O=C(O)C(OOCc1ccccc1)C(OOCc1ccccc1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 3/20 0.56
SLC1A3 P43003 2/20 0.56
SLC1A2 P43004 2/20 0.56
KMT2A Q03164 2/20 0.56
CYP1A2 P05177 2/20 0.56
MEN1 O00255 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
ALDH1A1 P00352 4/20 0.47
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TSHR P16473 3/20 0.43
SRR Q9GZT4 2/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10472894 1.00 SLC1A1 (0.56) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
SCHEMBL7603543 0.86 SLC1A1 (0.47) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
SCHEMBL1419749 0.81 ALDH1A1 (0.48) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
SCHEMBL9533527 0.80 L3MBTL1 (0.51) KMT2AMEN1ALDH1A1MAPK1L3MBTL1
SCHEMBL418322 0.79 SLC1A3 (0.76) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
SCHEMBL1953602 0.79 SLC1A3 (0.76) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
SCHEMBL852209 0.79 SLC1A3 (0.76) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
SCHEMBL8992078 0.79 SLC1A1 (0.41) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2
Bicarbonate SCHEMBL9066694 0.78 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1MAPK1L3MBTL1
Water SCHEMBL30419716 0.78 SLC1A3 (0.73) SLC1A1SLC1A3SLC1A2KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951051-A2 SPIROHYDANTOIN TRICYCLIC CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2008-08-06 EP disclosed
WO-2007061694-A2 SPIROHYDANTOIN TRICYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-05-31 WO disclosed
US-4251539-A HYPOTENSIVE AGENTS, ANTIARRHYTHMIA AGENTS BASF AKTIENGESELLSCHAFT (DE) 1981-02-17 US disclosed