SCHEMBL4962604

SCHEMBL4962604

CCC(O)(CC)Cc1csc(NS(=O)(=O)c2ccc(F)c(Cl)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.49
MEN1 O00255 7/20 0.47
POLB P06746 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
AGTR1 P30556 1/20 0.41
KDM1A O60341 1/20 0.41
PABPC1 P11940 1/20 0.41
SCN1A P35498 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN8A Q9UQD0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963088 0.85 KMT2A (0.63) KMT2AMEN1POLBALDH1A1PKM
SCHEMBL4964034 0.83 L3MBTL1 (0.53) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL4964626 0.82 KMT2A (0.50) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL4964602 0.81 KMT2A (0.43) KMT2AMEN1POLBALDH1A1PKM
SCHEMBL4963670 0.80 KMT2A (0.78) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL4967543 0.80 KMT2A (0.42) KMT2AMEN1POLBALDH1A1PKM
SCHEMBL4963626 0.76 KMT2A (0.48) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL4964890 0.76 HSD11B1 (0.66) KMT2AMEN1POLBALDH1A1CYP2C9
SCHEMBL4962933 0.76 KMO (0.43) KMT2AALDH1A1MAPTPKMSCN1A
SCHEMBL4962582 0.76 HSD11B1 (0.41) KMT2AALDH1A1MAPTPKMSCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed