SCHEMBL4963375

SCHEMBL4963375

[CH2][C@@H]1COc2cccc(-c3ccc(OCC)cc3C)c2O1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
NPC1 O15118 2/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
USP2 O75604 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAOB P27338 1/20 0.34
GRM5 P41594 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR1A P08908 2/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
FFAR1 O14842 1/20 0.34
ADRB2 P07550 3/20 0.33
ADRB1 P08588 3/20 0.33
ADRB3 P13945 2/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4959966 0.86 TSHR (0.41) TSHRNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL4963282 0.74 POLB (0.41) TSHRSMN1; SMN2ALDH1A1GAAMAOB
SCHEMBL8225830 0.71 AQP1 (0.39) TSHRKDM4EALDH1A1MAOBGRM5
SCHEMBL8210618 0.70 PRKAB2 (0.40) NPC1RAB9AKDM4EMAOBGRM5
SCHEMBL3218254 0.69 PRKAB2 (0.33) SMN1; SMN2KDM4EALDH1A1GAAUSP2
SCHEMBL3197092 0.69 PRKAB2 (0.33) SMN1; SMN2KDM4EALDH1A1GAAUSP2
SCHEMBL3220054 0.69 PRKAB2 (0.33) SMN1; SMN2KDM4EALDH1A1GAAUSP2
SCHEMBL6106691 0.69 CA2 (0.38) RAB9AGAAFFAR1
SCHEMBL4962940 0.68 ADRA2A (0.40) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL14364274 0.66 MAPT (0.45) TSHRSMN1; SMN2KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871759-A1 BENZODIOXANE AND BENZODIOXOLANE DERIVATIVES AND USES THEREOF Wyeth a Corporation of the State of Delaware (US) 2008-01-02 EP disclosed
WO-2006116158-A1 BENZODIOXANE AND BENZODIOXOLANE DERIVATIVES AND USES THEREOF WYETH (US) 2006-11-02 WO disclosed