SCHEMBL4963448

SCHEMBL4963448

CCCCc1cc(C#N)ccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.40
TSHR P16473 2/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP19A1 P11511 6/20 0.39
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
IDO1 P14902 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7219031 0.89 KDM4E (0.49) MBOAT4TSHRKDM4ELMNACYP3A4
SCHEMBL3242600 0.82 CYP1A2 (0.44) MBOAT4CTSSCTSKCCNCCDK8
SCHEMBL11365491 0.79 CCNC (0.53) LMNACYP3A4CYP19A1CCNCCDK8
SCHEMBL17843154 0.79 CCNC (0.41) MBOAT4TSHRKDM4ELMNACYP3A4
SCHEMBL3870198 0.79 CCNC (0.40) MBOAT4TSHRKDM4ELMNACYP3A4
SCHEMBL3869976 0.79 CCNC (0.40) MBOAT4LMNACYP19A1CCNCCDK8
SCHEMBL7219740 0.78 NOS2 (0.46) TSHRHSD17B10CYP19A1CTSSCTSK
SCHEMBL22637777 0.78 MBOAT4 (0.39) MBOAT4CYP19A1CCNCCDK8GAK
SCHEMBL15778536 0.77 KDM5A (0.61) CYP19A1
SCHEMBL6560564 0.76 KDM4E (0.44) TSHRKDM4ELMNACYP3A4GABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008030408-A2 PROTEOMIMETIC COMPOUNDS AS INHIBITORS OF THE INTERACTION OF A NUCLEAR RECEPTOR WITH COACTIVATOR PEPTIDES YALE UNIVERSITY (US) 2008-03-13 WO disclosed
US-6603007-B1 Intermediates in the fields of pharmaceuticals, agrichemicals, ligands, silver halide photosensitive materials, liquid crystals, surfactants, electrophotography and organic electroluminescence SANKIO CHEMICAL CO., LTD. (JP) 2003-08-05 US disclosed
EP-1231207-A1 NOVEL BIPYRIDYL DERIVATIVES Sankio Chemical Co., Ltd. (JP) 2002-08-14 EP disclosed