SCHEMBL4964673

SCHEMBL4964673

CCC(O)(CC)c1csc(NS(=O)(=O)c2cccc(Br)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 10/20 0.53
MAOA P21397 6/20 0.53
HSD17B2 P37059 1/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
EDNRB P24530 2/20 0.43
EDNRA P25101 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4966790 0.87 KDM1A (0.45) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4966051 0.84 KDM1A (0.60) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4964018 0.84 ALDH1A1 (0.47) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4962685 0.84 MEN1 (0.60) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4965945 0.83 GLO1 (0.48) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4964152 0.83 CA1 (0.40) KDM1AMAOAHSD17B2MEN1KMT2A
SCHEMBL4965545 0.82 KMT2A (0.46) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4966328 0.82 CA1 (0.44) KDM1AMAOAHSD17B2MEN1KMT2A
SCHEMBL4965281 0.82 MEN1 (0.64) KDM1AMAOAMEN1KMT2AALDH1A1
SCHEMBL4964537 0.81 MEN1 (0.43) KDM1AMAOAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed