SCHEMBL4964869

SCHEMBL4964869

O=C1[N]c2c(cc(Cc3ccccc3)cc2OC2CNC2)N1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.41
HTR6 P50406 4/20 0.39
HTR2C P28335 3/20 0.39
HTR2B P41595 3/20 0.39
HTR1A P08908 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HRH1 P35367 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4964772 0.89 HRH1 (0.51) HRH1
Hydrochloric Acid SCHEMBL4964910 0.83 KIT (0.39) SLC6A4
SCHEMBL4964913 0.82 SCN9A (0.37) HTR2BHRH1
SCHEMBL4964731 0.78 KIT (0.42) SLC6A4SLC6A2SLC6A3HRH1
SCHEMBL4966050 0.76 GABRA1 (0.38) SLC6A4HTR1ASLC6A2SLC6A3HRH1
SCHEMBL4964287 0.74 HRH1 (0.43) SLC6A4HRH1
SCHEMBL4963979 0.73 IDH1 (0.44)
SCHEMBL4963958 0.73 HRH1 (0.49) HRH1
SCHEMBL4966480 0.71 TAAR1 (0.46) SLC6A4HTR6HTR2CHTR1ASLC6A2
SCHEMBL4966731 0.68 TAAR1 (0.41) HTR6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP claimed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO claimed