SCHEMBL4963979

SCHEMBL4963979

O=C1[N]c2c(O)cc(Cc3ccccc3)cc2N1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.44
HNF4A P41235 1/20 0.39
BCL2 P10415 1/20 0.39
BCL2L1 Q07817 1/20 0.39
MPO P05164 1/20 0.38
PARP1 P09874 3/20 0.38
DAO P14920 1/20 0.38
PTPN1 P18031 3/20 0.37
PTPN2 P17706 1/20 0.37
PTPN6 P29350 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
CALM1 P0DP23 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4966731 0.76 TAAR1 (0.41) PTPN1PTPN2PTPN6
SCHEMBL4966480 0.74 TAAR1 (0.46)
SCHEMBL4964869 0.73 SLC6A4 (0.41)
SCHEMBL4964287 0.73 HRH1 (0.43)
SCHEMBL4966050 0.72 GABRA1 (0.38)
SCHEMBL4963958 0.72 HRH1 (0.49)
SCHEMBL4964772 0.72 HRH1 (0.51)
Hydrochloric Acid SCHEMBL4964910 0.71 KIT (0.39) DAO
SCHEMBL6230711 0.69 MEN1 (0.37) PARP1DAOALOX5
SCHEMBL278794 0.67 IDH1 (0.65) IDH1HNF4ABCL2BCL2L1MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed