SCHEMBL4965155

SCHEMBL4965155

CC(=O)Nc1ncc(Cc2cc(S(=O)(=O)N3CCCC(O)C3)sc2Br)s1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OGA O60502 13/20 0.43
OPRK1 P41145 1/20 0.42
LMNA P02545 3/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
PIK3CG P48736 1/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1237592 0.83 OGA (0.45) OGAOPRK1LMNAMAPTKMT2A
SCHEMBL1235241 0.76 PIK3CG (0.52) LMNAMAPTKMT2APIK3CGUSP2
SCHEMBL4672859 0.73 LMNA (0.53) OGALMNAMAPTKMT2AMEN1
SCHEMBL4960521 0.72 LMNA (0.45) OGAOPRK1LMNAMAPTKMT2A
SCHEMBL4964973 0.72 LMNA (0.47) OGALMNAMAPTKMT2AMEN1
SCHEMBL4959701 0.72 LMNA (0.47) OGALMNAMAPTKMT2AMEN1
SCHEMBL4960772 0.70 LMNA (0.45) LMNAMAPTKMT2AMEN1PIK3CG
SCHEMBL1236816 0.70 PIK3CG (0.47) LMNAKMT2APIK3CGUSP2TSHR
SCHEMBL4962537 0.69 LMNA (0.44) OGALMNAMAPTKMT2AMEN1
SCHEMBL1235188 0.67 PIK3CG (0.51) LMNAKMT2APIK3CGUSP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885716-A1 THIAZOLE DERIVATIVES AND USE THEREOF Laboratoires Serono SA (CH) 2008-02-13 EP disclosed
WO-2006125803-A1 THIAZOLE DERIVATIVES AND USE THEREOF LABORATOIRES SERONO S.A. (CH) 2006-11-30 WO disclosed