SCHEMBL4966468

SCHEMBL4966468

CCC(O)(CC)Cc1csc(NS(=O)(=O)c2ccc(CCCCN3CCOCC3)cc2C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.39
HSD11B1 P28845 4/20 0.37
NMT1 P30419 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
LMNA P02545 2/20 0.36
TSHR P16473 1/20 0.36
HSD17B1 P14061 2/20 0.36
HSD17B2 P37059 2/20 0.36
ALDH1A1 P00352 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
UBE2N P61088 1/20 0.35
POLB P06746 3/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LSS P48449 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963210 0.98 TRPV4 (0.40) TRPV4HSD11B1NMT1CNR1CNR2
SCHEMBL4965593 0.92 NMT1 (0.44) TRPV4HSD11B1NMT1CNR1CNR2
SCHEMBL4964100 0.90 NMT1 (0.47) TRPV4HSD11B1NMT1CNR1CNR2
SCHEMBL4964132 0.87 ROCK1 (0.42) TRPV4LMNATSHRALDH1A1SIGMAR1
SCHEMBL4965583 0.84 NPC1 (0.43) TRPV4HSD11B1ALDH1A1UBE2NMEN1
SCHEMBL4966824 0.79 NPC1 (0.42) TRPV4HSD11B1LMNATSHRALDH1A1
SCHEMBL4966984 0.78 HDAC3 (0.48) LMNATSHRALDH1A1SIGMAR1SMN1; SMN2
SCHEMBL4964824 0.77 EPHX2 (0.49) TRPV4TSHRALDH1A1KDM4ESMN1; SMN2
SCHEMBL4963626 0.76 KMT2A (0.48) HSD11B1LMNAHSD17B1HSD17B2ALDH1A1
SCHEMBL4962705 0.76 HSD11B1 (0.42) HSD11B1NMT1HSD17B1HSD17B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed