SCHEMBL4965760

SCHEMBL4965760

CCCCCn1nc(-c2ccccc2)[nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 4/20 0.48
SMPD1 P17405 1/20 0.47
MEN1 O00255 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
KMT2A Q03164 2/20 0.45
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
NR1H3 Q13133 1/20 0.44
ADORA2A P29274 3/20 0.44
MAPT P10636 1/20 0.43
MPO P05164 1/20 0.43
PDE5A O76074 1/20 0.42
CNR1 P21554 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP3A4 P08684 1/20 0.42
SLC5A1 P13866 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12400717 0.83 ADORA2B (0.48) ADORA2BMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL7656600 0.75 ALDH1A1 (0.49) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL3265647 0.74 ATM (0.65) ADORA2BCYP1A2ADORA2AMAPTPDE5A
SCHEMBL4965756 0.71 MEN1 (0.50) ADORA2BMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL7654102 0.69 ADORA2B (0.41) ADORA2BMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8741444 0.68 HTR2A (0.41) ADORA2BMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL5497681 0.68 CYP2C19 (0.44) SMPD1MEN1CYP1A2CYP2C9CYP2C19
SCHEMBL10419241 0.68 HCAR2 (0.35) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL15759808 0.67 BTK (0.46) ADORA2BMEN1CYP1A2KMT2AADORA2A
SCHEMBL13068443 0.67 BTK (0.46) ADORA2BMEN1CYP1A2KMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008106202-A1 THERAMUTEIN MODULATORS HOUSEY GERARD M (US) 2008-09-04 WO disclosed