SCHEMBL4965756

SCHEMBL4965756

CCCCCn1[nH]c(-c2ccccc2)nc1=O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ADORA2B P29275 4/20 0.45
TLR8 Q9NR97 2/20 0.43
CXCR2 P25025 1/20 0.42
ADORA2A P29274 3/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HSF1 Q00613 1/20 0.41
XDH P47989 1/20 0.40
PDE5A O76074 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656605 0.75 CXCR2 (0.67) CXCR2
SCHEMBL7649050 0.74 KDM4E (0.47) MEN1KMT2AADORA2BCXCR2ADORA2A
SCHEMBL4965760 0.71 ADORA2B (0.48) MEN1KMT2AADORA2BADORA2AKDM4E
SCHEMBL7654106 0.69 MGLL (0.44) MEN1KMT2AADORA2BCXCR2ADORA2A
SCHEMBL8741446 0.67 CXCR2 (0.47) MEN1KMT2AADORA2BCXCR2KDM4E
SCHEMBL7658198 0.67 KDM4E (0.44) MEN1KMT2AADORA2BCXCR2ADORA2A
SCHEMBL23400900 0.67 MEN1 (1.00) MEN1KMT2AADORA2BADORA2AKDM4E
SCHEMBL23398967 0.67 MEN1 (0.52) MEN1KMT2AADORA2BADORA2AKDM4E
SCHEMBL7650665 0.66 KDM4E (0.64) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL5328859 0.66 PDE4A (0.43) KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008106202-A1 THERAMUTEIN MODULATORS HOUSEY GERARD M (US) 2008-09-04 WO disclosed