SCHEMBL4965823

SCHEMBL4965823

NC(=O)Oc1ccc2c(c1)CCc1cc(CNC3CCCCCCC3)ccc1O2

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HDAC1 Q13547 1/20 0.44
HRH3 Q9Y5N1 2/20 0.39
POLB P06746 2/20 0.39
MCHR1 Q99705 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
CHEK1 O14757 1/20 0.37
TSHR P16473 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC8A1 P32418 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963719 1.00 MEN1 (0.45) MEN1KMT2AHDAC1HRH3POLB
SCHEMBL4968562 0.86 HDAC6 (0.45) MEN1KMT2AHDAC1MCHR1ALDH1A1
SCHEMBL4966804 0.84 HDAC1 (0.52) MEN1KMT2AHDAC1HRH3POLB
SCHEMBL4964378 0.84 HDAC1 (0.52) MEN1KMT2AHDAC1HRH3POLB
SCHEMBL4966598 0.82 MCHR1 (0.41) MEN1KMT2APOLBMCHR1ALDH1A1
Trifluoroacetic Acid SCHEMBL4966249 0.81 HDAC6 (0.40) HDAC1POLBALDH1A1KDM4ESLC8A1
SCHEMBL4971525 0.77 OPRM1 (0.40) MEN1KMT2AHDAC1POLBALDH1A1
SCHEMBL4968023 0.77 OPRM1 (0.46) POLBMCHR1NPC1RAB9A
SCHEMBL4965638 0.76 OPRM1 (0.41) HDAC1HRH3SMN1; SMN2
SCHEMBL4965646 0.76 OPRM1 (0.41) MEN1KMT2AHDAC1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP claimed