SCHEMBL4968562

SCHEMBL4968562

NC(=O)Oc1ccc2c(c1)CCc1cc(CNCC3CCCCC3)ccc1O2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.45
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
MCHR1 Q99705 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36
SRC P12931 1/20 0.36
F2 P00734 1/20 0.36
PLG P00747 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4966249 0.93 HDAC6 (0.40) HDAC6OPRM1OPRD1OPRK1HDAC3
SCHEMBL4966598 0.90 MCHR1 (0.41) HDAC6OPRM1OPRD1OPRK1MCHR1
SCHEMBL4963719 0.86 MEN1 (0.45) HDAC1MCHR1SLC8A1KMT2AALDH1A1
SCHEMBL4965823 0.86 MEN1 (0.45) HDAC1MCHR1SLC8A1KMT2AALDH1A1
SCHEMBL5332629 0.84 OPRM1 (0.58) HDAC6OPRM1OPRD1OPRK1HDAC3
SCHEMBL4965887 0.84 OPRM1 (0.58) HDAC6OPRM1OPRD1OPRK1HDAC3
SCHEMBL4968023 0.82 OPRM1 (0.46) OPRM1OPRD1OPRK1MCHR1ITGB3
SCHEMBL4971525 0.81 OPRM1 (0.40) OPRM1OPRK1HDAC1SLC8A1KMT2A
SCHEMBL4965646 0.79 OPRM1 (0.41) OPRM1OPRD1OPRK1HDAC1PRSS1
SCHEMBL4965638 0.79 OPRM1 (0.41) OPRM1OPRD1OPRK1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP claimed