SCHEMBL4965638

SCHEMBL4965638

CCCCCNCc1ccc2c(c1)CCc1cc(OC(N)=O)ccc1O2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
SLC2A1 P11166 1/20 0.41
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
S1PR1 P21453 4/20 0.38
S1PR3 Q99500 4/20 0.38
S1PR2 O95136 3/20 0.38
LPAR2 Q9HBW0 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
LMNA P02545 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963457 0.99 SLC2A1 (0.42) OPRM1OPRD1OPRK1SLC2A1HRH4
SCHEMBL4967478 0.89 KDM4E (0.49) SLC2A1SMN1; SMN2LMNA
SCHEMBL4965138 0.89 MCHR1 (0.43) SLC2A1SMN1; SMN2HDAC3HDAC1HDAC2
SCHEMBL4966629 0.88 SLC2A1 (0.37) OPRM1OPRD1OPRK1SLC2A1S1PR1
SCHEMBL4966256 0.86 AURKA (0.35) SLC2A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4965633 0.86 OPRM1 (0.45) OPRM1OPRD1OPRK1S1PR1S1PR3
SCHEMBL4965646 0.85 OPRM1 (0.41) OPRM1OPRD1OPRK1SLC2A1SMN1; SMN2
SCHEMBL4965252 0.85 OPRM1 (0.41) OPRM1OPRD1OPRK1SLC2A1
Hydrochloric Acid SCHEMBL4965277 0.84 OPRM1 (0.41) OPRM1OPRD1OPRK1SMN1; SMN2CYP2D6
SCHEMBL4964364 0.84 OPRM1 (0.57) OPRM1OPRD1OPRK1HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP claimed