SCHEMBL4968023

SCHEMBL4968023

NC(=O)Oc1ccc2c(c1)CCc1cc(CNCCC3CCOCC3)ccc1O2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.46
OPRK1 P41145 2/20 0.46
OPRD1 P41143 1/20 0.46
MCHR1 Q99705 3/20 0.40
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
CHRM2 P08172 4/20 0.34
CHRM1 P11229 4/20 0.34
CHRM3 P20309 4/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
MAPT P10636 1/20 0.33
RYR2 Q92736 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4966598 0.92 MCHR1 (0.41) OPRM1OPRK1OPRD1MCHR1RAB9A
SCHEMBL4965903 0.85 OPRM1 (0.61) OPRM1OPRK1OPRD1MCHR1RAB9A
SCHEMBL4968054 0.83 PARP1 (0.43) POLBMAPT
SCHEMBL4968562 0.82 HDAC6 (0.45) OPRM1OPRK1OPRD1MCHR1ITGB3
SCHEMBL4965252 0.82 OPRM1 (0.41) OPRM1OPRK1OPRD1MCHR1RAB9A
SCHEMBL5668119 0.82 OPRM1 (0.53) OPRM1OPRK1OPRD1MCHR1RAB9A
SCHEMBL4966564 0.81 MEN1 (0.44) POLBMAPTKCNH2
SCHEMBL4965638 0.80 OPRM1 (0.41) OPRM1OPRK1OPRD1DRD2
SCHEMBL4965646 0.80 OPRM1 (0.41) OPRM1OPRK1OPRD1RAB9ANPC1
SCHEMBL4967478 0.80 KDM4E (0.49) MCHR1RAB9ANPC1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP claimed