SCHEMBL4966458

SCHEMBL4966458

CCC(O)(CC)c1csc(NS(=O)(=O)c2ccc3c(c2)N(C)CCO3)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.51
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
RECQL P46063 1/20 0.44
SCN9A Q15858 4/20 0.43
HDAC3 O15379 2/20 0.42
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC9 Q9UKV0 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42
HTR6 P50406 1/20 0.42
POLB P06746 1/20 0.42
KDM1A O60341 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963200 0.86 ALDH1A1 (0.55) PKMALDH1A1HTTKDM1AMAOA
SCHEMBL4964583 0.84 ALDH1A1 (0.50) PKMKMT2AALDH1A1HTTSCN9A
SCHEMBL4963573 0.83 KDM4E (0.51) PKMKMT2AALDH1A1HTTHDAC3
SCHEMBL4968653 0.82 GLO1 (0.48) PKMKMT2AALDH1A1HTTHDAC3
SCHEMBL4968749 0.77 SMN1; SMN2 (0.56) PKMKMT2AALDH1A1HTTRAB9A
SCHEMBL4965545 0.76 KMT2A (0.46) PKMKMT2AALDH1A1HTTPOLB
SCHEMBL4962685 0.75 MEN1 (0.60) PKMKMT2AALDH1A1HTTKDM1A
SCHEMBL4965824 0.75 KMT2A (0.51) PKMKMT2AALDH1A1POLBKDM1A
SCHEMBL4966790 0.74 KDM1A (0.45) KMT2AALDH1A1KDM1AMAOA
SCHEMBL4964738 0.74 KMT2A (0.50) PKMKMT2AALDH1A1HTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed