SCHEMBL4964100

SCHEMBL4964100

CCC(O)(CC)Cc1csc(NS(=O)(=O)c2ccc(CCCN3CCOCC3)cc2Cl)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NMT1 P30419 2/20 0.47
HSD11B1 P28845 4/20 0.43
HSD17B1 P14061 2/20 0.39
HSD17B2 P37059 2/20 0.39
KMT2A Q03164 3/20 0.38
TRPV4 Q9HBA0 1/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
SIGMAR1 Q99720 2/20 0.38
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
ALDH1A1 P00352 2/20 0.36
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965593 0.98 NMT1 (0.44) NMT1HSD11B1HSD17B1HSD17B2KMT2A
SCHEMBL4963210 0.92 TRPV4 (0.40) NMT1HSD11B1HSD17B1HSD17B2KMT2A
SCHEMBL4966468 0.90 TRPV4 (0.39) NMT1HSD11B1HSD17B1HSD17B2KMT2A
SCHEMBL4965636 0.83 HSD11B1 (0.43) NMT1HSD11B1HSD17B1HSD17B2KMT2A
SCHEMBL4962705 0.83 HSD11B1 (0.42) NMT1HSD11B1HSD17B1HSD17B2KMT2A
SCHEMBL4964132 0.81 ROCK1 (0.42) TRPV4SIGMAR1LMNATSHRALDH1A1
SCHEMBL4962582 0.81 HSD11B1 (0.41) HSD11B1KMT2ATRPV4ALDH1A1PDK1
SCHEMBL4965583 0.79 NPC1 (0.43) HSD11B1KMT2ATRPV4MEN1ALDH1A1
SCHEMBL4965266 0.78 HSD11B1 (0.44) HSD11B1KMT2ATRPV4SIGMAR1LMNA
SCHEMBL4962933 0.78 KMO (0.43) HSD11B1KMT2AALDH1A1PDK1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed