SCHEMBL4967808

SCHEMBL4967808

Cn1cnc(CNCCCN(Cc2ccc3c(c2)OCO3)C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 8/20 0.51
NOS1 P29475 6/20 0.51
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
APOBEC3A P31941 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
TSHR P16473 2/20 0.41
USP2 O75604 1/20 0.40
LTA4H P09960 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3564374 0.88 NOS2 (0.48) NOS2NOS1KDM4EALDH1A1SMN1; SMN2
SCHEMBL4971539 0.78 ALDH1A1 (0.54) KDM4EALDH1A1SMN1; SMN2GAANPSR1
SCHEMBL4969501 0.78 ALDH1A1 (0.49) KDM4EALDH1A1SMN1; SMN2GAANPSR1
SCHEMBL4974818 0.75 ALDH1A1 (0.53) KDM4EALDH1A1SMN1; SMN2GAANPSR1
SCHEMBL4969568 0.74 NOS1 (0.54) NOS2NOS1ALDH1A1SMN1; SMN2GAA
SCHEMBL4967815 0.73 ALDH1A1 (0.43) NOS2NOS1KDM4EALDH1A1SMN1; SMN2
SCHEMBL15703671 0.72 CALM1 (0.49) NOS2NOS1KDM4ETSHR
SCHEMBL3561504 0.70 TSHR (0.53) ALDH1A1SMN1; SMN2GAANPSR1TSHR
Hydrochloric Acid SCHEMBL8844093 0.69 HPGD (0.45) ALDH1A1SMN1; SMN2GAATSHRMEN1
SCHEMBL3558567 0.69 SMN1; SMN2 (0.44) NOS2NOS1KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954695-A1 NOVEL METHOD OF PREPARATION OF 5-CHLORO-3-IMIDAZOL-1-YL-[1,2,4]THIADIAZOLE AND (3-IMIDAZOL-1-YL-[1,2,4]THIADIAZOL-5-YL)-DIALKYL-AMINES Kalypsys, Inc. (US) 2008-08-13 EP disclosed
WO-2007062411-A1 NOVEL METHOD OF PREPARATION OF 5-CHLORO-3-IMIDAZOL-1-YL-[1,2,4]THIADIAZOLE AND (3-IMIDAZOL-1-YL-[1,2,4]THIADIAZOL-5-YL)-DIALKYL-AMINES KALYPSYS, INC. (US) 2007-05-31 WO disclosed