SCHEMBL4973138

SCHEMBL4973138

C#CCN(C)C1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ADH1C P00326 2/20 0.37
ADH1A P07327 2/20 0.37
KDM4E B2RXH2 1/20 0.36
ABCB11 O95342 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
AR P10275 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
PDE4A P27815 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740408 0.77 ADH1A (0.41) HRH4HRH3ADH1CADH1AKDM4E
SCHEMBL7742694 0.77 ADH1A (0.41) HRH4HRH3ADH1CADH1AKDM4E
SCHEMBL1582838 0.76 ADH1A (0.31) ADH1CADH1ACYP2D6SLC6A2SLC6A4
SCHEMBL14146643 0.75 MAOA (0.41) MAOAMAOB
SCHEMBL4520995 0.74 HRH4 (0.38) HRH4HRH3ADH1CADH1AKDM4E
SCHEMBL7139255 0.74 ADH1A (0.39) ADH1CADH1AKDM4ESIGMAR1ALDH1A1
SCHEMBL13296390 0.74 HRH3 (0.39) HRH4HRH3ADH1CADH1AKDM4E
SCHEMBL15600812 0.73 HRH4 (0.37) HRH4HRH3ADH1CADH1AKDM4E
SCHEMBL7447366 0.72 ADH1C (0.38) ADH1CADH1A
SCHEMBL25934757 0.72 HRH4 (0.34) HRH4HRH3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753723-B1 SUBSTITUTED QUINOLINE DERIVATIVES AS MITOTIC KINESIN INHIBITORS NOVARTIS VACCINES & DIAGNOSTIC (US) 2008-08-13 EP claimed
CN-1210250-C Benzene derivatives, preparation method and pharmaceutical compositions containing same SANOFI SYNTHELABO (FR) 2005-07-13 CN disclosed
US-6482986-B1 Benzene derivatives, preparation method and pharmaceutical compositions containing same SANOFI-SYNTHELABO (FR) 2002-11-19 US disclosed
CN-1355782-A Benzene derivatives, preparation method and pharmaceutical compositions containing same SANOFI SYNTHELABO (FR) 2002-06-26 CN disclosed
EP-1192122-A1 BENZENE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2002-04-03 EP disclosed
WO-2000076953-A1 BENZENE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2000-12-21 WO disclosed
US-4088772-A TRANQUILIZERS, ANALGESICS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-05-09 US disclosed
US-4077977-A Ethenoanthracenes E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-03-07 US disclosed
US-4076830-A TRANQUILIZERS, ANALGESICS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-02-28 US disclosed