SCHEMBL4973263

SCHEMBL4973263

COc1cccc(B(OB(O)c2ccc(Cl)cc2Cl)OB(O)c2ccc(Cl)cc2Cl)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.36
TTR P02766 2/20 0.36
ORAI1 Q96D31 1/20 0.36
ORAI2 Q96SN7 1/20 0.36
ORAI3 Q9BRQ5 1/20 0.36
ACHE P22303 2/20 0.34
MAPT P10636 4/20 0.33
KMT2A Q03164 4/20 0.33
MEN1 O00255 3/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 3/20 0.33
BCHE P06276 1/20 0.33
ERN1 O75460 1/20 0.33
GAA P10253 1/20 0.33
NR3C1 P04150 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4973256 0.85 ENPP2 (0.45) ENPP2TTRORAI1ORAI2ORAI3
SCHEMBL29427098 0.71 ENPP2 (0.63) ENPP2ORAI1ORAI2ORAI3MAPT
SCHEMBL15701857 0.71 TSHR (0.41) TTRMAPTKMT2AMEN1CYP3A4
SCHEMBL126401 0.71 ENPP2 (0.63) ENPP2ORAI1ORAI2ORAI3MAPT
SCHEMBL23077788 0.70 ENPP2 (0.45) ENPP2ORAI1ORAI2ORAI3ACHE
SCHEMBL7772580 0.68 KDM4E (0.50) ENPP2ORAI1ORAI2ORAI3MAPT
SCHEMBL19204646 0.65 TRPV4 (0.44) ENPP2TTRORAI1ORAI2ORAI3
SCHEMBL29644544 0.65 ENPP2 (0.52) ENPP2TTRORAI1ORAI2ORAI3
SCHEMBL385535 0.65 ENPP2 (0.52) ENPP2TTRORAI1ORAI2ORAI3
SCHEMBL1728265 0.64 CA12 (0.46) MAPTKDM4ECYP3A4ALOX15LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979335-A2 THIAZOLES AS 11 BETA-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2008-10-15 EP disclosed
WO-2007082808-A2 THIAZOLES AS 11 BETA-HSD1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-07-26 WO disclosed