SCHEMBL4978322

SCHEMBL4978322

N=C(NC(=O)COCC(=O)O)NC(=O)COCC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
CTH P32929 1/20 0.33
CBS P35520 1/20 0.33
THPO P40225 1/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
THRB P10828 1/20 0.32
PTGS1 P23219 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4472021 0.90 TSHR (0.33) TSHRCTHCBSTHPOPOLB
SCHEMBL4467707 0.83 TSHR (0.36) TSHRCTHCBSTHPOPOLB
SCHEMBL4977502 0.81 TSHR (0.37) TSHRCTHCBSTHPOPOLB
SCHEMBL4977113 0.77 TSHR (0.35) TSHRCTHCBSTHPOPOLB
SCHEMBL4472825 0.77 TSHR (0.39) TSHRCTHCBSTHPOPOLB
SCHEMBL4479756 0.76 TAS2R38 (0.39) TSHRCTHCBSTHPOPOLB
SCHEMBL4488898 0.76 KDM4E (0.34) TSHRCTHCBSTHPOPOLB
SCHEMBL26928 0.74
SCHEMBL11406963 0.73 FOLH1 (0.46) TSHRCTHCBSTHPOPOLB
SCHEMBL4478714 0.72 ALDH1A1 (0.33) TSHRCTHCBSTHPOPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685114-B1 ANTIBACTERIAL AND/OR ANTIPROTOZOAL NITROIMIDAZOLE DERIVATIVE COMPOUNDS WITH UREASE INHIBITOR ACTIVITY, PROCESS FOR PREPARING THESE COMPOUNDS AND USE IN PHARMACEUTICAL COMPOSITIONS AND MEDICINES. EMS SA (BR) 2008-10-15 EP claimed