SCHEMBL4478714

SCHEMBL4478714

O=C(O)COCC(=O)NC(=S)NO

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.33
KDM4E B2RXH2 3/20 0.33
TSHR P16473 2/20 0.33
KDM6B O15054 1/20 0.32
KDM5C P41229 1/20 0.32
FOLH1 Q04609 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
PHF8 Q9UPP1 1/20 0.32
KDM2A Q9Y2K7 1/20 0.32
MAPT P10636 5/20 0.32
POLB P06746 2/20 0.32
KMT2A Q03164 3/20 0.31
MEN1 O00255 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
THRB P10828 1/20 0.30
CRHBP P24387 1/20 0.30
CRHR2 Q13324 1/20 0.30
APOBEC3G Q9HC16 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
CTH P32929 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4977113 0.90 TSHR (0.35) ALDH1A1KDM4ETSHRMAPTPOLB
SCHEMBL4479756 0.79 TAS2R38 (0.39) ALDH1A1TSHRPOLBKMT2AL3MBTL1
SCHEMBL4488898 0.79 KDM4E (0.34) ALDH1A1KDM4ETSHRKDM6BKDM5C
SCHEMBL11406963 0.78 FOLH1 (0.46) KDM4ETSHRKDM6BKDM5CFOLH1
SCHEMBL4977502 0.76 TSHR (0.37) ALDH1A1TSHRMAPTPOLBKMT2A
SCHEMBL4472021 0.76 TSHR (0.33) ALDH1A1KDM4ETSHRKDM6BKDM5C
SCHEMBL4472825 0.72 TSHR (0.39) ALDH1A1TSHRPOLBKMT2AMEN1
SCHEMBL4978322 0.72 TSHR (0.35) ALDH1A1TSHRPOLBKMT2AL3MBTL1
SCHEMBL4975649 0.72 PHF8 (0.58) ALDH1A1KDM4EKDM6BKDM5CFOLH1
SCHEMBL4976250 0.72 FAAH (0.41) ALDH1A1KDM4ETSHRMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7608724-B2 2-(2-Methyl-5-nitro-1H-imidazol-1-yl)ethyl 4-[(aminocarbonothioyl)amino]-4-oxobutanoate;potententiation; anaerobic/ aerobic microoraganisms; grampositive,gramnegative bacteria; Campylobacter; respiratory system disorders; paraciticides; nontoxic; enzymers/hydrolases/;enzyme inhibitors EMS S.A. (BR) 2009-10-27 US claimed
EP-1685114-B1 ANTIBACTERIAL AND/OR ANTIPROTOZOAL NITROIMIDAZOLE DERIVATIVE COMPOUNDS WITH UREASE INHIBITOR ACTIVITY, PROCESS FOR PREPARING THESE COMPOUNDS AND USE IN PHARMACEUTICAL COMPOSITIONS AND MEDICINES. EMS SA (BR) 2008-10-15 EP claimed